Target Details
UniProt ACP04585
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 2,623
  • Clinical molecules 3
  • Avg pChEMBL 7.89
Top Co-occurrence Targets
Active Molecules (2,623)
InChIKey pChEMBL Type Targets Clinical
ULRNZWUMNJXISM 11.2 Ki 2
JOOIRGLUJVFIDO 11.0 Ki 2
VRSJYTMZDYBQTL 11.0 Ki 2
YSTMEPTXAKTZGG 11.0 Ki 2
NIGQODFLJMCYDF 11.0 Ki 2
NLVWCIHYQHCPFO 11.0 Ki 2
IWHMDIMNPYWHLJ 10.9 Ki 2
NVANLDBYIPHGQE 10.9 Ki 2
WCWRSOYUXMDNSR 10.9 Ki 2
LPGGYDYQUYLLOU 10.9 Ki 3
VBXNXLBIEHWXSR 10.9 IC50 2
BOSLDRMHSGQVEF 10.8 Ki 2
AFVXCMZTRNKQLP 10.8 IC50 2
LFGJUVNTHXGQFQ 10.8 Ki 2
MZJFSOKHVVULFM 10.8 Ki 2
NIEAPINYNLFWMC 10.8 Ki 2
OMGSSZKVQUJYTF 10.8 Ki 2
WBEKUEKRXIUAHQ 10.8 Ki 2
YJOUONBJMOBWJG 10.8 Ki 2
ZZEQQJBEFIZMSK 10.8 Ki 2
GRHZLQBPAJAHDM 10.8 Ki 3
KJHKTHWMRKYKJE 10.8 Ki 4
AKSONJGXCNANNF 10.7 Ki 2
BLPYBPRQGPFMDB 10.7 Ki 2
GUUBIMLFZZKWRX 10.7 Ki 2
GYVMEIFMNCTCMZ 10.7 Ki 3
JIICMIOQFYIENG 10.7 Ki 2
LBKKHTKXYVYCDI 10.7 Ki 2
MZBJXKMJVLOTIB 10.7 Ki 2
PPZYUYUJMYWIHM 10.7 Ki 2
WENVZQWSDCKTAH 10.7 Ki 3
GNPYXBMOZFIQNG 10.7 Ki 2
JZLATAYRZNKODI 10.7 Ki 2
KNPACJDWGFHMIF 10.7 Ki 2
OIIBJJOGEBWRPK 10.7 Ki 2
SDULFQOGIXPXRD 10.7 Ki 2
SMPFVGOGVVEABT 10.7 Ki 2
XYUHJAIPECDEBR 10.7 Ki 2
CGEJBZXGNPASAG 10.7 Ki 3
WZSNGBIAZKDCIX 10.7 Ki 2
YWYRHXOIDGHGTC 10.7 Ki 2
HCKQNDUSXFAVMA 10.7 Ki 2
DTARGNCRAXTWIW 10.6 Ki 2
FJWVGEMWYQYGGB 10.6 Ki 2
LXMZTSYDUPYAMZ 10.6 Ki 2
ZMYUVMXCSCTAQG 10.6 Ki 2
DNHYOPVNRBAZMG 10.6 Ki 2
DRIQIEGYOOXTGG 10.6 Ki 2
FOEKUOOABOINMH 10.6 Ki 2
JDALSSGOBMTZEP 10.6 Ki 2
2D structure