Target Details
| UniProt AC | P04278 |
|---|---|
| Gene Symbol | SHBG |
| Protein Name | Sex hormone-binding globulin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00054 (Laminin_G_1) |
Summary
- Multi-target molecules 24
- Clinical molecules 4
- Avg pChEMBL 7.44
Active Molecules (24)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QADHLRWLCPCEKT
|
9.2 | Kd | 4 | — | |
NVKAWKQGWWIWPM
|
9.1 | IC50 | 5 | — | |
WWYNJERNGUHSAO
|
8.9 | Kd | 3 | — | |
CHNXZKVNWQUJIB
|
8.8 | Kd | 2 | — | |
MUMGGOZAMZWBJJ
|
8.5 | IC50 | 6 | — | |
GCKMFJBGXUYNAG
|
8.4 | Kd | 2 | — | |
POZRVZJJTULAOH
|
8.2 | Kd | 3 | — | |
DNXHEGUUPJUMQT
|
8.2 | Kd | 4 | — | |
VOXZDWNPVJITMN
|
8.1 | IC50 | 8 | — | |
VIKNJXKGJWUCNN
|
8.0 | Kd | 6 | Yes | |
AEMFNILZOJDQLW
|
7.5 | Kd | 6 | Yes | |
WHBHBVVOGNECLV
|
7.4 | Kd | 2 | — | |
ZESRJSPZRDMNHY
|
7.4 | Kd | 5 | — | |
DBPWSSGDRRHUNT
|
7.0 | Kd | 3 | — | |
RJKFOVLPORLFTN
|
6.9 | Kd | 10 | Yes | |
BFPYWIDHMRZLRN
|
6.8 | Kd | 10 | — | |
PROQIPRRNZUXQM
|
6.6 | Kd | 2 | — | |
LPYXTAPPNYMYOP
|
6.4 | Kd | 2 | — | |
OMFXVFTZEKFJBZ
|
6.3 | Kd | 4 | — | |
NPAGDVCDWIYMMC
|
6.3 | Kd | 2 | — | |
JYGXADMDTFJGBT
|
6.2 | Kd | 4 | — | |
PSGAAPLEWMOORI
|
6.2 | Kd | 11 | Yes | |
QGXBDMJGAMFCBF
|
6.2 | Kd | 2 | — | |
FTVWIRXFELQLPI
|
6.0 | Kd | 6 | — |