Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DLXBCJBMEVKPIX
|
7.3 | Ki | 9 | Yes | |
MEWQFKSUHJZGCA
|
7.3 | Ki | 4 | — | |
VDCNLLFWCBGVMM
|
7.3 | IC50 | 3 | — | |
YKQNBGVCIMLMLA
|
7.3 | Ki | 3 | — | |
GGQRUDKBZGUEAN
|
7.3 | IC50 | 2 | — | |
MOMZVCIJGACLFL
|
7.3 | IC50 | 2 | — | |
PDQVCFOQIMKRGZ
|
7.3 | IC50 | 3 | — | |
JJSZJRHRVRGDNH
|
7.3 | IC50 | 2 | — | |
VBGYFNUDIFNZRO
|
7.3 | Ki | 3 | — | |
AUIFRJWXYUNPPV
|
7.3 | IC50 | 2 | — | |
NOUXCOKPRXVTDP
|
7.3 | Ki | 3 | — | |
UZSAWQCKBUFFQD
|
7.3 | IC50 | 2 | — | |
NVKFRYWNCLQAGR
|
7.2 | Ki | 2 | — | |
BVXLAHSJXXSWFF
|
7.2 | IC50 | 2 | — | |
CTRKFGYVXQHNDJ
|
7.2 | IC50 | 2 | — | |
RXVVCKDZPLPROM
|
7.2 | IC50 | 2 | — | |
SWLSHPWYSWBPQE
|
7.2 | IC50 | 2 | — | |
AFQIBZSGVWHLSI
|
7.2 | IC50 | 2 | — | |
DUZBBWARHFOMBJ
|
7.2 | IC50 | 3 | — | |
IXMWYDAQMMZUOZ
|
7.2 | IC50 | 2 | — | |
KGFMFEQQZNKWLP
|
7.2 | IC50 | 3 | — | |
LWYLVQVGWUQBSI
|
7.2 | Ki | 2 | — | |
XZKRNADKQRQVOR
|
7.2 | IC50 | 2 | — | |
ZDCRSQSGCDAAAC
|
7.2 | IC50 | 2 | — | |
CEDQCHHKNHJFKO
|
7.2 | IC50 | 2 | — | |
DBWRTNRVJFYFDM
|
7.2 | IC50 | 2 | — | |
JQMVFHXSBNJQRP
|
7.2 | IC50 | 2 | — | |
PZTMIXXVWUCYIR
|
7.2 | IC50 | 2 | — | |
BXRDIKRRETWSCY
|
7.2 | IC50 | 2 | — | |
HSLFOYFJYRSLKF
|
7.2 | IC50 | 3 | — | |
TZSWJUXVIXDAFP
|
7.2 | IC50 | 2 | — | |
DZIWDYAOHLYJGW
|
7.2 | IC50 | 2 | — | |
KYUGYVXBKPAWOH
|
7.2 | IC50 | 3 | — | |
GAUXDXUKQPFNPK
|
7.2 | IC50 | 6 | Yes | |
NSEYQHXUJJGSKW
|
7.2 | IC50 | 2 | — | |
RSVKCRGCARHPAC
|
7.1 | IC50 | 4 | — | |
XVYWAUINFAXEKA
|
7.1 | IC50 | 3 | — | |
DPAAYBADQOGZSY
|
7.1 | IC50 | 2 | — | |
RRDSVYGZMKNAFC
|
7.1 | IC50 | 2 | — | |
FXSCCOANJPANKE
|
7.1 | IC50 | 3 | — | |
NIJXJFCGNYEYSG
|
7.1 | IC50 | 2 | — | |
WJEDKJKCQOZDNI
|
7.1 | IC50 | 3 | — | |
XFLYEUSUDVNPKL
|
7.1 | Ki | 2 | — | |
KDMGOYHSUFIUAT
|
7.1 | IC50 | 2 | — | |
QQFIDVOPZHXZPF
|
7.1 | IC50 | 3 | — | |
WNRXXFMGMKLIHP
|
7.1 | IC50 | 5 | Yes | |
XYAPBFRUZQERGJ
|
7.1 | IC50 | 2 | — | |
BDYFDDGUXXUNJN
|
7.1 | IC50 | 5 | Yes | |
JLMKYNGLORSHHP
|
7.1 | IC50 | 2 | — | |
WGGMBWMYJSVPSG
|
7.1 | IC50 | 3 | — |