Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAEZOVLEAHIZGN
|
7.6 | IC50 | 2 | — | |
ZJHROHSTVJKUKT
|
7.6 | IC50 | 2 | — | |
KIXSJEJHLVMNMZ
|
7.6 | IC50 | 2 | — | |
UPKAUNVEGRFAII
|
7.6 | IC50 | 2 | — | |
UTPNUAIWPWLJEC
|
7.6 | IC50 | 4 | — | |
QKBURCBWLIXXPH
|
7.6 | Ki | 2 | — | |
WISJIBWIQKICSR
|
7.6 | Ki | 2 | — | |
LCTFQUGGLDHXTH
|
7.5 | IC50 | 3 | — | |
XCCRMYVOJIFMED
|
7.5 | IC50 | 3 | — | |
IRZVQRHERMOSEM
|
7.5 | Ki | 2 | — | |
KNEYKCUMUCBZNB
|
7.5 | IC50 | 3 | — | |
GAKWAQHHESGFAA
|
7.5 | IC50 | 3 | — | |
HGSACWBRJAQDIP
|
7.5 | IC50 | 2 | — | |
RJKFOVLPORLFTN
|
7.5 | Ki | 10 | Yes | |
SXIDZLMPGLSSSR
|
7.5 | IC50 | 4 | — | |
NWSIDHCBAFDSKX
|
7.5 | Ki | 2 | — | |
RASBRABSHNFWAA
|
7.5 | IC50 | 2 | — | |
LXMSZDCAJNLERA
|
7.5 | Ki | 6 | Yes | |
QAIBFISDVFSRKN
|
7.5 | IC50 | 2 | — | |
NNEGFNICKYKFDF
|
7.5 | IC50 | 2 | — | |
QHSJNOYFBNQNIZ
|
7.5 | IC50 | 2 | — | |
VPBRSFFMKTUJNN
|
7.5 | IC50 | 2 | — | |
XOSVCJKDUIUUIB
|
7.5 | Ki | 2 | — | |
DBPWSSGDRRHUNT
|
7.5 | IC50 | 3 | — | |
HJOUYAMEBCDGKK
|
7.5 | IC50 | 2 | — | |
MWIXIWILHMYRGD
|
7.5 | IC50 | 3 | — | |
WWKUDAJCCSNRRV
|
7.5 | IC50 | 3 | — | |
XYFAXIKXGILQET
|
7.5 | IC50 | 2 | — | |
TVKQINGZQAQVCA
|
7.5 | IC50 | 2 | — | |
SSAMEZHVGWGDGH
|
7.4 | IC50 | 3 | — | |
CVFDJBVNXZCLBL
|
7.4 | IC50 | 2 | — | |
YRAUBPBLFNFPPH
|
7.4 | IC50 | 2 | — | |
FMZKGKLLLCYGJW
|
7.4 | IC50 | 3 | — | |
GHRAAOQUALWOAH
|
7.4 | IC50 | 2 | — | |
GOUMJTGDXMAQKS
|
7.4 | IC50 | 2 | — | |
QOZZBCZFOZCNQK
|
7.4 | IC50 | 3 | — | |
VPBRSFFMKTUJNN
|
7.4 | IC50 | 2 | — | |
PSGAAPLEWMOORI
|
7.4 | Ki | 2 | — | |
AZKXBAPRQCXHRZ
|
7.4 | IC50 | 2 | — | |
HFWXCPFGOCGJDK
|
7.4 | IC50 | 3 | — | |
OIXUDXUFFGADIZ
|
7.3 | IC50 | 2 | — | |
XDAWAGMTCJTDDV
|
7.3 | IC50 | 2 | — | |
UDQPQRQPOLSCKG
|
7.3 | IC50 | 2 | — | |
UKKKPJSCGQJZAT
|
7.3 | IC50 | 2 | — | |
ANPFZNKOHNLVIS
|
7.3 | IC50 | 2 | — | |
IMDWWFBCGVBAMW
|
7.3 | IC50 | 2 | — | |
JRIIXIXSRVUNTB
|
7.3 | IC50 | 2 | — | |
IMTGEDOKMRCXLE
|
7.3 | Ki | 6 | Yes | |
BTEQZWJLBYEBLQ
|
7.3 | Ki | 4 | — | |
CERMKIOTMWNAGM
|
7.3 | Ki | 2 | — |