Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UPXAYCYCDXAKMG
|
7.7 | Ki | 2 | — | |
VEASGQCTQWVLOL
|
7.7 | IC50 | 2 | — | |
VPGLREFJYMSJHR
|
7.7 | IC50 | 2 | — | |
KVPALVACWJUWHG
|
7.7 | IC50 | 6 | Yes | |
OTKZWGJLFLAVTD
|
7.7 | IC50 | 2 | — | |
GJXAQWRUPWTIBX
|
7.7 | IC50 | 2 | — | |
QPLQDYDXYCUKKE
|
7.7 | IC50 | 3 | — | |
CCMNCWDOPDWHKL
|
7.7 | IC50 | 2 | — | |
HMYGXGUMESBWOB
|
7.7 | IC50 | 2 | — | |
LQAJJWMXZBDMAC
|
7.7 | IC50 | 2 | — | |
QAJXXFBIGIATMT
|
7.7 | Ki | 2 | — | |
RINQMJSFPWHRTD
|
7.7 | Ki | 2 | — | |
XZOCWBJVVFJEFU
|
7.7 | IC50 | 2 | — | |
ZXXGFBBNJBARSN
|
7.7 | IC50 | 2 | — | |
ZZWNDPPQMABJJG
|
7.7 | IC50 | 3 | — | |
HYZGNFIJTUJTBY
|
7.7 | IC50 | 2 | — | |
NHIKVVXPLBWTNX
|
7.7 | IC50 | 3 | — | |
PHCCLYMMALQRTG
|
7.7 | IC50 | 2 | — | |
QFXLFIGPPAXZQQ
|
7.7 | IC50 | 2 | — | |
QHIXHFRNTAVAPK
|
7.7 | IC50 | 2 | — | |
UGJGTPGLSLQCPP
|
7.7 | IC50 | 3 | — | |
WFIFLFARTXGDFP
|
7.7 | IC50 | 2 | — | |
HINCRROTVFUICG
|
7.7 | IC50 | 3 | — | |
LUMRHKVOXMIPGU
|
7.7 | IC50 | 2 | — | |
ARAFJNZXJVLHDR
|
7.7 | IC50 | 3 | — | |
BFWRCRIDNKRGTD
|
7.7 | IC50 | 2 | — | |
IYIBSFQMWALFFX
|
7.7 | Ki | 2 | — | |
YWPNXVQAAHGWCZ
|
7.7 | IC50 | 2 | — | |
ZREYWBOITVVPOZ
|
7.7 | IC50 | 3 | — | |
ZRFGZMFRRNHMLW
|
7.7 | IC50 | 2 | — | |
BDZYLNZLEGRWAZ
|
7.7 | IC50 | 2 | — | |
PKGWJFNRGGGBJB
|
7.7 | IC50 | 3 | — | |
KDVSANSBFHATHQ
|
7.6 | IC50 | 2 | — | |
PEEQAQFTZGENDO
|
7.6 | IC50 | 2 | — | |
ROGXRBIZXSSLJN
|
7.6 | IC50 | 2 | — | |
YXGACPVGUQXDFZ
|
7.6 | IC50 | 2 | — | |
BCWFWNBNYVPLRF
|
7.6 | IC50 | 3 | — | |
DCRMRSLJFCGKKG
|
7.6 | IC50 | 2 | — | |
FLBVZAVMHFNOKV
|
7.6 | IC50 | 2 | — | |
VWCZQZNHWPQZGT
|
7.6 | IC50 | 3 | — | |
WANIDIGFXJFFEL
|
7.6 | Ki | 2 | — | |
MKBMFZOEUDKVGZ
|
7.6 | IC50 | 2 | — | |
MTJXQXWQRBOMIO
|
7.6 | IC50 | 2 | — | |
NXRVYSZNJVQSEI
|
7.6 | IC50 | 2 | — | |
PUCKHCPITYMJIM
|
7.6 | IC50 | 2 | — | |
RFDCXOHZVYCSJT
|
7.6 | Ki | 2 | — | |
XLVWWNSBFIWDGB
|
7.6 | IC50 | 2 | — | |
YXQPDNYJXVGIES
|
7.6 | Ki | 2 | — | |
YKFHUVOJZGWRDY
|
7.6 | IC50 | 2 | — | |
JYGXADMDTFJGBT
|
7.6 | Ki | 4 | — |