Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BAOUXBDVAPNGRU
|
7.9 | IC50 | 2 | — | |
HXJYKDIOBRNHTQ
|
7.9 | IC50 | 2 | — | |
RLNRYNADPTVFSB
|
7.9 | Ki | 2 | — | |
SGSLRJUNARVKFS
|
7.9 | IC50 | 3 | — | |
SIMVLEKLLFIFBJ
|
7.9 | IC50 | 2 | — | |
ADHVTOAGYGEFSM
|
7.9 | IC50 | 2 | — | |
LIYOMQNHCSVUSQ
|
7.9 | IC50 | 2 | — | |
QLZJETYFHQVNRB
|
7.9 | IC50 | 2 | — | |
JNJSRSUVKCYZLN
|
7.9 | IC50 | 2 | — | |
OKMFMKSZIXQMRJ
|
7.9 | IC50 | 2 | — | |
WPGAOHWZNCMFLY
|
7.9 | IC50 | 2 | — | |
OZBSREXZWADXQE
|
7.9 | IC50 | 3 | — | |
PBRBWYQRHGSGKO
|
7.9 | IC50 | 2 | — | |
PSGAAPLEWMOORI
|
7.9 | Ki | 11 | Yes | |
RZCOQAQHAZHWEB
|
7.9 | IC50 | 3 | — | |
UUIWYLMDKKQBJQ
|
7.9 | IC50 | 3 | — | |
CFDUSNZVLMAHPE
|
7.9 | IC50 | 3 | — | |
SMYUZCJLGBMSME
|
7.9 | IC50 | 3 | — | |
DIAWBONHWJRWKZ
|
7.9 | IC50 | 2 | — | |
NNTHLQVZGURUAX
|
7.9 | IC50 | 3 | — | |
QTOKABCAHAKYAS
|
7.9 | IC50 | 2 | — | |
KJUOEYJRZUJJLM
|
7.8 | IC50 | 3 | — | |
SSFWXDSRZJERKU
|
7.8 | Ki | 2 | — | |
YJGVMLPVUAXIQN
|
7.8 | IC50 | 19 | — | |
YTKAYWYQPDHXNV
|
7.8 | IC50 | 3 | — | |
NNWXOVXANQHVST
|
7.8 | IC50 | 2 | — | |
BQZKKRYIQPCEKF
|
7.8 | IC50 | 2 | — | |
CPXLOFOGNURDFC
|
7.8 | IC50 | 3 | — | |
FGWOYLFOCSKTSC
|
7.8 | IC50 | 2 | — | |
IDCRMONFSJJBMN
|
7.8 | IC50 | 3 | — | |
RBUVZQPMAIWWCG
|
7.8 | IC50 | 2 | — | |
ZCEACWHBZXPKIT
|
7.8 | IC50 | 2 | — | |
DHMLTYBVPKCCCQ
|
7.8 | IC50 | 2 | — | |
DQCNRZPBBUYZOQ
|
7.8 | IC50 | 2 | — | |
PFUXODWITQFWRK
|
7.8 | IC50 | 2 | — | |
STJWTSUWXXKJNZ
|
7.8 | IC50 | 2 | — | |
VPIGGHQZYNIAQH
|
7.8 | IC50 | 2 | — | |
YFJZCMOHVUUOJJ
|
7.8 | IC50 | 2 | — | |
BBICQKYRAXECKV
|
7.8 | IC50 | 3 | — | |
ONOSXGJCDWPVFI
|
7.8 | IC50 | 2 | — | |
ORHHWJMIJCSUTC
|
7.8 | IC50 | 2 | — | |
VWTXAIVZMCQYKU
|
7.8 | IC50 | 3 | — | |
VVCVRVUPFSJFRH
|
7.8 | IC50 | 3 | — | |
AAJNWJFLYOFHIB
|
7.8 | IC50 | 3 | — | |
FEKIYUBTGQLEBI
|
7.8 | IC50 | 3 | — | |
ULOAOMMDFZMTER
|
7.8 | IC50 | 3 | — | |
UYBJISPAOAQTKQ
|
7.8 | IC50 | 2 | — | |
OWWJZAKLVDXCMD
|
7.7 | IC50 | 2 | — | |
QYGXPNCCWFGVRU
|
7.7 | Ki | 2 | — | |
UDDUGXMYFCMHJO
|
7.7 | IC50 | 3 | — |