Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VGCGSAUUQCQDAY
|
8.1 | IC50 | 3 | — | |
YXBSHEFOZZFYPO
|
8.1 | IC50 | 2 | — | |
YROYMPDJQKBNTG
|
8.1 | IC50 | 3 | — | |
PAUIGLFJCJDVFW
|
8.1 | IC50 | 2 | — | |
SFFRJYDGTHMNDH
|
8.1 | IC50 | 3 | — | |
HINCRROTVFUICG
|
8.1 | IC50 | 3 | — | |
USMFOMVHIKQVEN
|
8.1 | IC50 | 3 | — | |
CEOIQIXVRWVLBN
|
8.1 | IC50 | 3 | — | |
JQDUVTPGLRBCNA
|
8.1 | IC50 | 3 | — | |
LBBVZEVHJCWQLW
|
8.1 | IC50 | 2 | — | |
PDCRQOSNBYFZJI
|
8.1 | IC50 | 2 | — | |
LMAFSLWCXOQARP
|
8.1 | IC50 | 4 | — | |
OMIMAFBBRNJDDU
|
8.1 | IC50 | 3 | — | |
SUBXROOMJNLXRP
|
8.1 | Ki | 2 | — | |
UCLMIPKAOVLOQS
|
8.1 | IC50 | 2 | — | |
ZILACWFNZFWDAS
|
8.1 | IC50 | 3 | — | |
LFLARVMSGCQYSZ
|
8.0 | IC50 | 2 | — | |
UHIXENGVNOWISA
|
8.0 | IC50 | 2 | — | |
ANIOYQXTAMMUKZ
|
8.0 | Ki | 2 | — | |
DORQSUNHACTGLQ
|
8.0 | IC50 | 3 | — | |
LCDCPIOGHJGDBP
|
8.0 | IC50 | 2 | — | |
OHDDNRZGDGYKBR
|
8.0 | IC50 | 2 | — | |
ZAINQQRFGATLID
|
8.0 | IC50 | 4 | — | |
CCCIJQPRIXGQOE
|
8.0 | Ki | 4 | — | |
GUJAUKQZCIPIBV
|
8.0 | IC50 | 4 | Yes | |
OUXFXJUDVPDIII
|
8.0 | IC50 | 2 | — | |
QOSRQKJZZAEYCI
|
8.0 | IC50 | 2 | — | |
BBQPRPRCQIFLIO
|
8.0 | Ki | 2 | — | |
BYVDCSLCMPQTKD
|
8.0 | Ki | 2 | — | |
FNAPHRONLYQVOG
|
8.0 | IC50 | 2 | — | |
GKQWMOXIBZCMDJ
|
8.0 | IC50 | 3 | — | |
GWBHDCFCUBNVKR
|
8.0 | IC50 | 2 | — | |
JKPOACVGQYPLBU
|
8.0 | IC50 | 3 | — | |
PVYTWCNJUWKUOG
|
8.0 | IC50 | 3 | — | |
SGPHLLUCLSONGK
|
8.0 | IC50 | 2 | — | |
YBIHCFXAMSLIHT
|
8.0 | IC50 | 2 | — | |
YSJVBSSZEGNKMZ
|
8.0 | IC50 | 2 | — | |
ZVCDNODZUJDLPU
|
8.0 | IC50 | 2 | — | |
ABDAGDDZOUDCKI
|
8.0 | IC50 | 2 | — | |
WFSBONJXUAXVJH
|
8.0 | IC50 | 3 | — | |
ALDWINSGSURGLP
|
8.0 | IC50 | 3 | — | |
MPLPTTLNPDVGGI
|
8.0 | IC50 | 2 | — | |
NYAOFNPTQGNQKM
|
8.0 | IC50 | 2 | — | |
NZKHJRBHEWBIFL
|
8.0 | IC50 | 3 | — | |
QOSRQKJZZAEYCI
|
8.0 | IC50 | 2 | — | |
VRZVKIJRJRBQJT
|
8.0 | IC50 | 4 | — | |
MXEOXTXWJGNBGH
|
7.9 | IC50 | 2 | — | |
OJVZKFXAMCVCKM
|
7.9 | IC50 | 2 | — | |
QDMKBJCCHCGTOQ
|
7.9 | IC50 | 2 | — | |
FFJPGJNSRNWRSX
|
7.9 | IC50 | 2 | — |