Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PHUOGFXDMSBGIK
|
8.3 | IC50 | 2 | — | |
GDJKXOLGMVNOGF
|
8.2 | IC50 | 3 | — | |
DCDROSDZJJENGM
|
8.2 | IC50 | 3 | — | |
QGCIAWJCSRYRFH
|
8.2 | Ki | 2 | — | |
DJRNAIGSFHOUFL
|
8.2 | IC50 | 2 | — | |
KJOQLFMPAVEWLJ
|
8.2 | IC50 | 3 | — | |
WUXTURZHMMFRPK
|
8.2 | IC50 | 3 | — | |
NLPNUYHHRWOSGM
|
8.2 | IC50 | 4 | — | |
OYHQTRCZCQLKPX
|
8.2 | IC50 | 2 | — | |
QSDGRHKNICEVHX
|
8.2 | IC50 | 3 | — | |
RSMAEJMIEPTWJC
|
8.2 | IC50 | 2 | — | |
YTMMXBWUMWUPPN
|
8.2 | Ki | 2 | — | |
ZOUVODOOOFQPOC
|
8.2 | IC50 | 2 | — | |
MIAURGNSNSBTNK
|
8.2 | Ki | 4 | — | |
WFQCSOVOMJIJSZ
|
8.2 | IC50 | 2 | — | |
ABDAGDDZOUDCKI
|
8.2 | IC50 | 2 | — | |
BQDLKNZJOSLJEM
|
8.2 | Ki | 2 | — | |
DJRNAIGSFHOUFL
|
8.2 | IC50 | 2 | — | |
JQDUVTPGLRBCNA
|
8.2 | IC50 | 3 | — | |
JTNNQTQMGYMRGO
|
8.2 | IC50 | 3 | — | |
OIGNJSKKLXVSLS
|
8.2 | IC50 | 7 | — | |
YUENOOALVDTBKW
|
8.2 | IC50 | 2 | — | |
SLKURXRZHJOZOD
|
8.2 | Ki | 2 | — | |
XFFATDFCPKLQRT
|
8.2 | Ki | 2 | — | |
QOOAVFNQEWFRQY
|
8.2 | Ki | 2 | — | |
DXVZGTRLQAZISS
|
8.2 | IC50 | 2 | — | |
GCKMJAVBEKTJOI
|
8.2 | IC50 | 2 | — | |
IFFNOGXSDVOOPK
|
8.2 | IC50 | 2 | — | |
LVZOQUMLGOHFGL
|
8.2 | IC50 | 3 | — | |
OTNBHAGJVFDFBS
|
8.2 | Ki | 2 | — | |
PCEQNBCVZPRGRR
|
8.2 | IC50 | 3 | — | |
ADHVTOAGYGEFSM
|
8.1 | IC50 | 2 | — | |
CFDUSNZVLMAHPE
|
8.1 | IC50 | 3 | — | |
MDMKCVXYKPOLIM
|
8.1 | Ki | 2 | — | |
NOUXCOKPRXVTDP
|
8.1 | Ki | 4 | — | |
DJDDNTUYFUVZIC
|
8.1 | IC50 | 2 | — | |
KSINXTGJLYCZIP
|
8.1 | Ki | 2 | — | |
HKLWSBIHHHYTLH
|
8.1 | IC50 | 2 | — | |
PCGWJSDLFYYVRR
|
8.1 | IC50 | 2 | — | |
PDEYZVGOCYDQJF
|
8.1 | IC50 | 3 | — | |
QTOKABCAHAKYAS
|
8.1 | IC50 | 3 | — | |
XXWVLLGWBXOMHQ
|
8.1 | IC50 | 2 | — | |
AZYGKDQZZHOKOM
|
8.1 | IC50 | 2 | — | |
CIIHIZKWQHRFRR
|
8.1 | IC50 | 2 | — | |
GIBZLWRPPUSMTC
|
8.1 | IC50 | 4 | — | |
ICFLHQGITDWVMH
|
8.1 | Ki | 2 | — | |
MHWZNBBELRMCAO
|
8.1 | IC50 | 3 | — | |
OUCNRPREOGLYEL
|
8.1 | Ki | 2 | — | |
QEMGULFBAZGYKI
|
8.1 | IC50 | 2 | — | |
RCRRMTBHOFTNFS
|
8.1 | IC50 | 2 | — |