Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LTVDMZKEGDEQLE
|
8.6 | Ki | 2 | — | |
NMWIJNGJMPMFQG
|
8.6 | IC50 | 2 | — | |
DQMJJYWWVJPLDX
|
8.6 | Ki | 2 | — | |
KAFURNBTIHQXCB
|
8.6 | IC50 | 2 | — | |
MPEPSOPXQDGEHP
|
8.6 | IC50 | 2 | — | |
CVNFMOXXWTZVDU
|
8.5 | IC50 | 2 | — | |
UREBDLICKHMUKA
|
8.5 | IC50 | 13 | — | |
VYJSUSIGTRGXQC
|
8.5 | IC50 | 3 | — | |
YUMWHZCQHQAPAQ
|
8.5 | IC50 | 3 | — | |
ZDRUXXZVOLZIBA
|
8.5 | Ki | 2 | — | |
LKQMULLPLYLIGW
|
8.5 | IC50 | 3 | — | |
LKQMULLPLYLIGW
|
8.5 | IC50 | 3 | — | |
JFUAWXPBHXKZGA
|
8.5 | IC50 | 2 | — | |
MXEOXTXWJGNBGH
|
8.5 | IC50 | 2 | — | |
HUPZROPFBRSFDW
|
8.5 | IC50 | 2 | — | |
KPKCYUMBFMYREG
|
8.5 | IC50 | 3 | — | |
RITZPFDVXSENFR
|
8.5 | IC50 | 2 | — | |
VWFKACUYWYZVSW
|
8.5 | IC50 | 3 | — | |
UMKDQHBGTUYJCV
|
8.4 | IC50 | 2 | — | |
HAJBHFSMKOWEHU
|
8.4 | IC50 | 2 | — | |
QURQZQPYRJKKHS
|
8.4 | IC50 | 2 | — | |
RWLAOUIUIWXAOY
|
8.4 | Ki | 2 | — | |
JPEBLWKHCCIJKH
|
8.4 | IC50 | 2 | — | |
YGMWYZPIFDQGCI
|
8.4 | IC50 | 3 | — | |
DKFBPHVUBSXDJB
|
8.4 | IC50 | 3 | — | |
FBHBBILQSLGKPC
|
8.4 | Ki | 2 | — | |
NGLPZZZUWGVILU
|
8.4 | IC50 | 2 | — | |
RGMOSYPQLNCAFJ
|
8.4 | IC50 | 3 | — | |
VKVZOFDGLCTSKW
|
8.4 | Ki | 2 | — | |
VQMSYLLYQOARPD
|
8.4 | IC50 | 3 | — | |
ZANAAVXGSNLYBQ
|
8.4 | IC50 | 2 | — | |
PMRWVBCWVGHOPT
|
8.4 | IC50 | 2 | — | |
CPUIRDMVUBPAPK
|
8.4 | Ki | 3 | — | |
HHJSGMINRSKVLO
|
8.3 | IC50 | 3 | — | |
PYHAWYQXRVXAHX
|
8.3 | IC50 | 4 | — | |
VDSMZEJGVOMCGQ
|
8.3 | IC50 | 2 | — | |
FAZOJHMTURPXLD
|
8.3 | IC50 | 2 | — | |
JRZWVYSKNVMDLP
|
8.3 | IC50 | 3 | — | |
NAKVZBYNDIOTLA
|
8.3 | IC50 | 3 | — | |
XNVXVNJRQLVPBF
|
8.3 | IC50 | 2 | — | |
UCWWMUPWYRSGBY
|
8.3 | IC50 | 2 | — | |
SEVGDNHYESBDRZ
|
8.3 | IC50 | 2 | — | |
NLDACKJWSTTYSC
|
8.3 | IC50 | 2 | — | |
DOSZIFWFKFJGQL
|
8.3 | IC50 | 3 | — | |
XFFATDFCPKLQRT
|
8.3 | Ki | 2 | — | |
CAVTYMQSFAIXRJ
|
8.3 | IC50 | 4 | — | |
AJAOWKDQDBTLKO
|
8.3 | IC50 | 2 | — | |
KSRJOQNNZWTUHC
|
8.3 | Ki | 2 | — | |
MIPUTBSSNQTOCB
|
8.3 | Ki | 2 | — | |
SAVAEFOXNWPFKB
|
8.3 | IC50 | 3 | — |