Target Details
UniProt ACP04150
Gene SymbolNR3C1
Protein NameGlucocorticoid receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 632
  • Clinical molecules 32
  • Avg pChEMBL 7.64
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (632)
InChIKey pChEMBL Type Targets Clinical
BEOADSCNJSAOSW 8.9 Ki 2
QBUKAFSEUHGMMX 8.9 Ki 2
ZITUOTORLGBDOZ 8.9 IC50 2
MRSXXYFEMRTFDC 8.9 Ki 2
BLPNJKOYOIDEJJ 8.9 IC50 2
QYEYUIJWYCBKBG 8.9 Ki 2
AJJYMQGHGPINNM 8.8 Ki 2
ATJGOPJRRWGHHL 8.8 IC50 4
LEOCLJZACQHETJ 8.8 IC50 4
MJQKPIOTILTXNU 8.8 Ki 2
DSMDXILQYZQPHU 8.8 IC50 2
DYJSODVHTVCXIA 8.8 Ki 4
NREZDYQUMMSPNC 8.8 Ki 2
RVDUZNHKCJRYQY 8.8 Ki 2
VOVIALXJUBGFJZ 8.8 IC50 4
YFJZCMOHVUUOJJ 8.8 IC50 3
JSNLQEVTILZGHC 8.8 IC50 2
QKTUOSGGPMYODZ 8.8 Ki 2
MATZYFFMBFOOKH 8.8 Ki 2
DORQSUNHACTGLQ 8.8 IC50 3
CFZKPYJJGYQRFD 8.7 IC50 2
MFAGIEMFDDDLMT 8.7 IC50 3
IBEIVQBULJKLFB 8.7 IC50 2
UXGUYYJUKZKENF 8.7 Ki 2
AKMUGEXFTSZYPE 8.7 Ki 2
DLHJAQJQFLHXNZ 8.7 IC50 2
FTNKKFZQMNEADX 8.7 IC50 2
HKLWSBIHHHYTLH 8.7 IC50 3
QGPHIACZTUTSAR 8.7 IC50 2
RXEIQMFFHIVGLD 8.7 IC50 3
UUGJKSUOOIUEHL 8.7 Ki 2
VQXYALIFGGOXRU 8.7 Ki 2
XEDXLCMFJIIBOV 8.7 IC50 2
PFBJOLPYJDUPPW 8.7 IC50 2
LPVOSIGKKGTQCK 8.7 Ki 2
ORSBFWQUUWUENG 8.7 IC50 2
CUNSDNZRZMUTPA 8.7 Ki 2
VKNDUDKNPQIQIQ 8.7 Ki 3
CRODFMXMGHZTCT 8.6 Ki 2
VKYPRKNSJRILPH 8.6 Ki 2
ACYYHAZVNHMRMQ 8.6 Ki 4
JZDXQIACRWWJNM 8.6 IC50 2
QFWHAFOCMOQSHC 8.6 IC50 3
QWKSNMYGEFJJIU 8.6 Ki 2
KXMVPYRKURWIPA 8.6 IC50 4
NFAZOJQFTSWUIF 8.6 Ki 2
NMIXBOUDRDWICA 8.6 IC50 3
OAYLSAHITBROEB 8.6 IC50 2
USLSTEHVCOVPEK 8.6 IC50 3
KLTYQAJNDLZNSD 8.6 IC50 2
2D structure