Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQGIWZOYDNHCSJ
|
6.2 | IC50 | 2 | — | |
BVSCKUSMKCQTFI
|
6.1 | IC50 | 2 | — | |
UAXYYPCBGHLJKQ
|
6.1 | Ki | 3 | — | |
DRUKCDBJSKTKTR
|
6.1 | IC50 | 2 | — | |
JAPBAKGEKZXGRM
|
6.1 | IC50 | 3 | — | |
OSHWKQSKIVSROR
|
6.1 | IC50 | 2 | — | |
BFPYWIDHMRZLRN
|
6.1 | Ki | 10 | — | |
CJZROCCAPJVVQO
|
6.1 | IC50 | 3 | — | |
QFRVNOIAPBNRJM
|
6.1 | Ki | 2 | — | |
ACXANRVNFDEJLV
|
6.1 | Ki | 2 | — | |
GCKMFJBGXUYNAG
|
6.1 | Ki | 2 | — | |
QWPDOAPBJDUXDW
|
6.1 | IC50 | 2 | — | |
AHBGXQDJONQGOL
|
6.1 | IC50 | 2 | — | |
FQYNXWLDJCLBQP
|
6.1 | Ki | 3 | — | |
MFVGPPNQHPWGHH
|
6.1 | IC50 | 2 | — | |
QDBUCXMBHJMGCN
|
6.0 | IC50 | 4 | — | |
ZWGPOLYPUOBDPY
|
6.0 | IC50 | 2 | — | |
FOPLNUAISVOILB
|
6.0 | Ki | 3 | — | |
QXSLSLICSJPAFZ
|
6.0 | Ki | 2 | — | |
LSQKEQHYMWDEPS
|
6.0 | Ki | 2 | — | |
BPLVBRPOOZNKHW
|
6.0 | IC50 | 2 | — | |
PKBIAUYNZMVJCB
|
6.0 | IC50 | 2 | — | |
CUIMAZBZRVOSOP
|
6.0 | Ki | 3 | — | |
FPFITAPEARIFHY
|
6.0 | IC50 | 2 | — | |
AXOMYVRKJFDZJX
|
6.0 | Ki | 2 | — | |
BURHGPHDEVGCEZ
|
6.0 | IC50 | 3 | — | |
FGCNFOXYZQLPMW
|
6.0 | IC50 | 3 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
IMGXWRKTVOMDLZ
|
6.0 | IC50 | 3 | — | |
KYWWJENKIMRJBI
|
6.0 | IC50 | 3 | — | |
QEYIPZOJYLGUHY
|
6.0 | IC50 | 2 | — | |
QWWNXNFWXOZGLJ
|
6.0 | IC50 | 3 | — |