Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IJTNKDPWHRABRX
|
6.5 | Ki | 2 | — | |
IMTXAMMYSYUYSB
|
6.5 | Ki | 2 | — | |
JKBQDIAWGDKQHW
|
6.5 | IC50 | 2 | — | |
PLOQCPGEMKIJBX
|
6.5 | Ki | 2 | — | |
WLEYQRHXERCYNY
|
6.5 | IC50 | 3 | — | |
FOPLNUAISVOILB
|
6.5 | Ki | 2 | — | |
DGELEWLFMTZTAW
|
6.5 | IC50 | 2 | — | |
GQEDWCRZISUBTM
|
6.5 | Ki | 2 | — | |
HGHRCZOIYJBGPL
|
6.5 | IC50 | 3 | — | |
JJBGOTRJBHAAQW
|
6.5 | IC50 | 2 | — | |
FLXKJKBDBACQDP
|
6.4 | IC50 | 2 | — | |
IDGIKWDCKXJAES
|
6.4 | Ki | 3 | — | |
YGYIVBNMBYBQGZ
|
6.4 | IC50 | 3 | — | |
HMBNPWKLPBPJMY
|
6.4 | IC50 | 3 | — | |
MIAURGNSNSBTNK
|
6.4 | Ki | 4 | — | |
CWXNSHLNBNLSSS
|
6.4 | IC50 | 3 | — | |
DQALECYZLFPXOQ
|
6.4 | IC50 | 2 | — | |
JJTJZAROTNIJSJ
|
6.4 | Ki | 2 | — | |
KJSHBZLXBZYVMR
|
6.4 | Ki | 3 | — | |
MEFYNCWNNHNHMN
|
6.4 | IC50 | 3 | — | |
PHKMDGYGCDKJEU
|
6.4 | IC50 | 2 | — | |
VKUBXLNVYQUCFV
|
6.4 | IC50 | 2 | — | |
QTOKABCAHAKYAS
|
6.4 | IC50 | 2 | — | |
IMONTRJLAWHYGT
|
6.4 | IC50 | 2 | — | |
CXFSVKGROITHRY
|
6.3 | Ki | 3 | — | |
HQVKFEYATUGVGI
|
6.3 | IC50 | 2 | — | |
YISCUJJPIJSXKK
|
6.3 | IC50 | 2 | — | |
AWPVKERKWQLOEG
|
6.3 | IC50 | 4 | Yes | |
FDFMYVGKENHMGM
|
6.3 | IC50 | 2 | — | |
UFSVWJLQUADLKJ
|
6.3 | IC50 | 2 | — | |
KDBXYNSMRDJJFO
|
6.3 | IC50 | 2 | — | |
ZEZOALAOUQCQQW
|
6.3 | IC50 | 3 | — | |
CXXWEXDTTVWKSJ
|
6.3 | IC50 | 2 | — | |
JIKFLEZNTIZKCI
|
6.3 | Ki | 4 | — | |
HKKAPCOJXICOAX
|
6.3 | Ki | 2 | — | |
NVKAWKQGWWIWPM
|
6.3 | IC50 | 5 | — | |
YXKBVHXOKVRRKO
|
6.2 | Ki | 6 | Yes | |
ISFPMZBOTSJQDY
|
6.2 | IC50 | 2 | — | |
NDBQYPUELRHJBZ
|
6.2 | IC50 | 2 | — | |
WSOYYBRZDOKCSB
|
6.2 | Ki | 2 | — | |
WWTZCUBJPLJNNS
|
6.2 | Ki | 2 | — | |
AXXQTTPUMYEBOV
|
6.2 | IC50 | 4 | — | |
DUKSLEMXBDETTE
|
6.2 | IC50 | 2 | — | |
CVQKNTTYZMQDMD
|
6.2 | Ki | 2 | — | |
DVIBYGTZNAJRGB
|
6.2 | IC50 | 2 | — | |
CZHIJMGMBQCQDA
|
6.2 | Ki | 3 | — | |
OCLPHOSZZDWUFZ
|
6.2 | Ki | 2 | — | |
WFOHHEVAQLCSFM
|
6.2 | IC50 | 3 | — | |
ZBHGJXVSUFQFPP
|
6.2 | IC50 | 3 | — | |
CLQBRBFJGFBWMS
|
6.2 | IC50 | 3 | — |