Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RQUXQDVRWLHMBG
|
6.8 | IC50 | 2 | — | |
RTYKMFMHRRYCIK
|
6.8 | Ki | 2 | — | |
WIMXURNPWBOQET
|
6.8 | Ki | 4 | — | |
ZQFNDBISEYQVRR
|
6.8 | IC50 | 2 | — | |
BRWFVMSKOCNHHI
|
6.8 | IC50 | 2 | — | |
DFZYMRBKXQWSTE
|
6.8 | IC50 | 2 | — | |
MIAURGNSNSBTNK
|
6.8 | Ki | 4 | — | |
BQFHIOXHOTZDCT
|
6.8 | Ki | 2 | — | |
JTYKTQGMYNYWGT
|
6.8 | IC50 | 2 | — | |
VRWXHHASXOUVMH
|
6.8 | IC50 | 2 | — | |
OFPJLMJVJSEKIP
|
6.7 | IC50 | 3 | — | |
KGVGNTCIQIYLQU
|
6.7 | IC50 | 9 | Yes | |
XYBAXMXTSMKKKQ
|
6.7 | IC50 | 2 | — | |
BXMUAQLRVCWTKG
|
6.7 | IC50 | 3 | — | |
FQYNXWLDJCLBQP
|
6.7 | Ki | 3 | — | |
OZGJGGGYYPKMDN
|
6.7 | IC50 | 3 | — | |
CBUBLNUCASPVJQ
|
6.7 | Ki | 2 | — | |
GCBGSMQYZCPYLB
|
6.7 | IC50 | 2 | — | |
MGDHDHQGYPSORD
|
6.7 | IC50 | 3 | — | |
MMQYPFTZXJAWGY
|
6.7 | IC50 | 5 | Yes | |
WDYCDBMOJVBUFD
|
6.7 | IC50 | 3 | — | |
IFNZOVIDIOXFMG
|
6.7 | IC50 | 2 | — | |
NPDSJEIIHNPHHF
|
6.7 | Ki | 2 | — | |
QCRMHUMUIWUQMT
|
6.7 | Ki | 3 | — | |
WIUDNDXMQHQJIL
|
6.7 | IC50 | 2 | — | |
WDXRGPWQVHZTQJ
|
6.7 | Ki | 5 | — | |
DAYFWNQOWUPASA
|
6.6 | IC50 | 2 | — | |
HTCMKQLSSZWFTP
|
6.6 | IC50 | 5 | Yes | |
HQGRCFOENHIIQG
|
6.6 | IC50 | 2 | — | |
KCVAVMXQQQXOLI
|
6.6 | IC50 | 6 | Yes | |
WDXRGPWQVHZTQJ
|
6.6 | Ki | 5 | — | |
XGBWGDGYTTWUIM
|
6.6 | Ki | 3 | — | |
FDWPXNLUFQNWMH
|
6.6 | Ki | 2 | — | |
FZORYLRILGENBG
|
6.6 | Ki | 3 | — | |
QXSLSLICSJPAFZ
|
6.6 | Ki | 3 | — | |
RFZAHUIHPLZLLA
|
6.6 | Ki | 9 | Yes | |
WDXRGPWQVHZTQJ
|
6.6 | Ki | 5 | — | |
ZVALABNDJZPNNC
|
6.6 | IC50 | 3 | — | |
FZORYLRILGENBG
|
6.6 | Ki | 2 | — | |
LVCVMYKRVFAVCM
|
6.6 | IC50 | 6 | Yes | |
UDYVQHLPMVKSOP
|
6.6 | Ki | 3 | — | |
DFZYMRBKXQWSTE
|
6.6 | IC50 | 3 | — | |
LIHLXWYJHXJFEM
|
6.6 | IC50 | 3 | — | |
LQJIEYFFKBLJFV
|
6.6 | IC50 | 3 | — | |
FDMHMFIRHWCKNN
|
6.5 | IC50 | 2 | — | |
OVIZCQBEPZRBDB
|
6.5 | IC50 | 3 | — | |
RTLRJRHSVSOAFD
|
6.5 | IC50 | 3 | — | |
VIKNJXKGJWUCNN
|
6.5 | IC50 | 6 | Yes | |
XLIGSXQYXJZZSL
|
6.5 | IC50 | 2 | — | |
HFQCJPQBQUZNQQ
|
6.5 | IC50 | 2 | — |