Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
POYMYRFGHYKMSL
|
7.1 | IC50 | 4 | — | |
WCWNFANFHMNQEP
|
7.1 | IC50 | 7 | Yes | |
MYDJWFCWWHPKCH
|
7.0 | IC50 | 6 | Yes | |
JXRAVTIDZDMHLO
|
7.0 | Ki | 4 | — | |
PVUYPBAPWIWFAJ
|
7.0 | IC50 | 2 | — | |
YPUGASLTKIAOPT
|
7.0 | IC50 | 6 | Yes | |
DZKSHTKHHHLSGZ
|
7.0 | IC50 | 3 | — | |
FFFOIRSYFQWGQH
|
7.0 | Ki | 2 | — | |
GJMNAFGEUJBOCE
|
7.0 | IC50 | 5 | Yes | |
KTOKJEZDHROXCU
|
7.0 | IC50 | 2 | — | |
RCZNQWQDJPJWMD
|
7.0 | IC50 | 3 | — | |
WWYNJERNGUHSAO
|
7.0 | IC50 | 3 | — | |
ZUOVTFWGFULART
|
7.0 | IC50 | 2 | — | |
NTYALJAURYTROE
|
7.0 | IC50 | 6 | Yes | |
POUMWPFDKBAVDE
|
7.0 | IC50 | 2 | — | |
UKLYTFISJSJGSO
|
7.0 | IC50 | 2 | — | |
JZFUUMIFIPVITG
|
7.0 | IC50 | 2 | — | |
AHCZZOJYVQVLQG
|
6.9 | IC50 | 3 | — | |
GWXSFBMSMRCBDS
|
6.9 | IC50 | 2 | — | |
URYARKSTCIJGME
|
6.9 | Ki | 3 | — | |
VKUBXLNVYQUCFV
|
6.9 | IC50 | 2 | — | |
WZBNEBURHZRFPI
|
6.9 | IC50 | 2 | — | |
IHUHWAUMFFURSJ
|
6.9 | IC50 | 2 | — | |
WZKWYTSJJZVJLU
|
6.9 | IC50 | 3 | — | |
DZATYSMEKYVDKI
|
6.9 | IC50 | 6 | Yes | |
IZUMHFDUSAWWQU
|
6.9 | IC50 | 2 | — | |
NVMGBEWNMCNKHG
|
6.9 | Ki | 2 | — | |
OPPYDCXBDREGJT
|
6.9 | IC50 | 4 | — | |
POJKNBHEJAUGMR
|
6.9 | Ki | 2 | — | |
RKFFHZQKHIMLAH
|
6.9 | IC50 | 2 | — | |
AZXWUJXCVIDGJV
|
6.9 | IC50 | 2 | — | |
NBYXOMZEWLMKJB
|
6.9 | Ki | 3 | — | |
DJRBZWVBECJRTM
|
6.9 | IC50 | 2 | — | |
OHLMRBMVXRKABN
|
6.9 | Ki | 2 | — | |
PUQSDJZESAQGQS
|
6.9 | IC50 | 2 | — | |
CHNXZKVNWQUJIB
|
6.8 | IC50 | 2 | — | |
WSGANSMSRKUENH
|
6.8 | IC50 | 2 | — | |
NTCBYBDADUSXSB
|
6.8 | IC50 | 9 | Yes | |
VQFLIHCSQSPSJT
|
6.8 | IC50 | 3 | — | |
WVCKFHDLPYAJOU
|
6.8 | IC50 | 5 | — | |
CTCHAYJBEBAVDT
|
6.8 | IC50 | 6 | Yes | |
DTIMQMAYRMJPRM
|
6.8 | IC50 | 2 | — | |
HDCJFWTUMAKTNA
|
6.8 | IC50 | 2 | — | |
NTXRXSSTKKNELF
|
6.8 | IC50 | 5 | Yes | |
UWFYSQMTEOIJJG
|
6.8 | IC50 | 3 | — | |
WOYXGESYPYMTAQ
|
6.8 | Ki | 2 | — | |
BEQGDWGTHMWLCN
|
6.8 | IC50 | 2 | — | |
IAUDUYJHOKBQLW
|
6.8 | IC50 | 6 | Yes | |
NKLKXXWOFGFVKN
|
6.8 | Ki | 2 | — | |
NVTFLQJKFXTAOZ
|
6.8 | Ki | 2 | — |