Target Details
| UniProt AC | P04150 |
|---|---|
| Gene Symbol | NR3C1 |
| Protein Name | Glucocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02155 (GCR) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 632
- Clinical molecules 32
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (632)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WMWTYOKRWGGJOA
|
10.1 | IC50 | 4 | — | |
CNOAOQSZNOTZLQ
|
10.0 | Ki | 2 | — | |
FHYZXPHRIMDEBV
|
10.0 | IC50 | 2 | — | |
NSUUUQRFPXZFLI
|
10.0 | Ki | 2 | — | |
UFZZMZCIWOEUKP
|
9.8 | Ki | 4 | — | |
UZNBZDTUBTWOBU
|
9.7 | IC50 | 4 | — | |
GHQUUJUZRHSGHN
|
9.6 | IC50 | 2 | — | |
UITKQZZSZUEHEA
|
9.6 | IC50 | 2 | — | |
LGTLOCBNEXITRB
|
9.6 | Ki | 4 | — | |
PHIKAOOZNGLKDI
|
9.6 | Ki | 4 | — | |
WFESRNFSHAPECN
|
9.5 | Ki | 4 | Yes | |
XKUDSVCPHSGCDL
|
9.5 | IC50 | 2 | — | |
VLRUOHNPKMZQHN
|
9.5 | IC50 | 2 | — | |
QQGISFDJEJMKIL
|
9.4 | IC50 | 3 | — | |
ZTKAFVSUBJCXFM
|
9.4 | Ki | 3 | — | |
IDEHKJXWAPTFBV
|
9.4 | IC50 | 2 | — | |
ALJARNPEIWWIOU
|
9.4 | IC50 | 2 | — | |
VYMKIBYWMBCPEZ
|
9.3 | IC50 | 2 | — | |
NVBRVAKHESDYFE
|
9.3 | IC50 | 2 | — | |
XTLUPLYDVHOHSW
|
9.3 | IC50 | 4 | — | |
XTULMSXFIHGYFS
|
9.3 | IC50 | 3 | — | |
ZWTCGJWGJMGWIM
|
9.3 | Ki | 3 | — | |
CYBZSWXWFMWSAP
|
9.2 | Ki | 2 | — | |
PWKJVVLBXRWXFQ
|
9.2 | IC50 | 2 | — | |
CZOFJQFQALBETE
|
9.2 | IC50 | 4 | — | |
KHLLMEXZTPDMCY
|
9.2 | IC50 | 3 | — | |
OTWADYHEAKBKQC
|
9.2 | IC50 | 4 | — | |
WDSPVCXWXOIFRA
|
9.2 | Ki | 2 | — | |
AWBMTFDCCHSMQU
|
9.2 | Ki | 2 | — | |
HLRQXZBFIYYNOH
|
9.2 | Ki | 3 | — | |
HQFHTXSVKRXPKT
|
9.2 | Ki | 2 | — | |
PCJNAMBTUJABGN
|
9.2 | Ki | 2 | — | |
WOFMFGQZHJDGCX
|
9.2 | Ki | 3 | — | |
XLHCDLVMCWZSEQ
|
9.2 | IC50 | 2 | — | |
KVBSKVDOWUOCJZ
|
9.1 | Ki | 2 | — | |
ZDCMJDVSSLHLLQ
|
9.1 | Ki | 9 | Yes | |
ZSMCHXGGQCKXMY
|
9.1 | Ki | 5 | Yes | |
KAAJYBMWABCTAG
|
9.1 | IC50 | 4 | — | |
VXOKHYHZXBLDSC
|
9.1 | IC50 | 4 | — | |
DPPNIDONMQTQMK
|
9.1 | IC50 | 3 | — | |
FDXWONUERKJVPB
|
9.1 | Ki | 2 | — | |
KNTPSJWEFWVLCP
|
9.1 | Ki | 2 | — | |
OSRXVTVKOPCOGY
|
9.1 | IC50 | 3 | — | |
UWFYSQMTEOIJJG
|
9.1 | IC50 | 2 | — | |
FOSHWESRGNRMBT
|
9.0 | Ki | 2 | — | |
CBGUOGMQLZIXBE
|
9.0 | IC50 | 3 | — | |
DUVQYORBVMIRPF
|
9.0 | IC50 | 3 | — | |
PNVTUJVNNJCYGM
|
9.0 | IC50 | 3 | — | |
RKZJWUOBFCJJTR
|
9.0 | Ki | 2 | — | |
MLZLXEBPLLEJSK
|
8.9 | IC50 | 2 | — |