Target Details
| UniProt AC | P04114 |
|---|---|
| Gene Symbol | APOB |
| Protein Name | Apolipoprotein B-100 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12491 (ApoB100_C) PF06448 (DUF1081) PF09172 (Vit_open_b-sht) PF01347 (Vitellogenin_N) |
Summary
- Multi-target molecules 47
- Clinical molecules 0
- Avg pChEMBL 8.38
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (47)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JKHYOWBRQRJSTQ
|
9.2 | IC50 | 2 | — | |
NXEKMMKJEQUKOX
|
9.1 | IC50 | 2 | — | |
MUSVRXWCIMGFPH
|
9.0 | IC50 | 2 | — | |
JXAAATVXBZVTFP
|
9.0 | IC50 | 2 | — | |
FNNZOYHEGGNTMW
|
8.9 | IC50 | 2 | — | |
SPCXYBUWDJJYRU
|
8.9 | IC50 | 2 | — | |
WOKRZDMTEXOXTC
|
8.8 | IC50 | 2 | — | |
MLJWCPIALKPLOS
|
8.8 | IC50 | 2 | — | |
NLYURQFDYAGQOK
|
8.8 | IC50 | 2 | — | |
VFQLHOJNCNGPIK
|
8.8 | IC50 | 3 | — | |
NGBACBJFDKYOER
|
8.7 | IC50 | 2 | — | |
PMXMADULYZHDGE
|
8.7 | IC50 | 2 | — | |
WYTALJCRYOJNIS
|
8.7 | IC50 | 2 | — | |
IECYXABIVIGSDE
|
8.7 | IC50 | 2 | — | |
XIPGMFZCORQMAY
|
8.7 | IC50 | 2 | — | |
DPKBSACUADFSQG
|
8.7 | IC50 | 2 | — | |
OLXBRQXHOJCVJV
|
8.7 | IC50 | 2 | — | |
QWPNUQHQVLSBQS
|
8.7 | IC50 | 2 | — | |
ZPLGGQUGKMCWQW
|
8.7 | IC50 | 2 | — | |
IPKSAVBBDPQPEF
|
8.6 | IC50 | 2 | — | |
KAVUYBYDHINKNE
|
8.6 | IC50 | 2 | — | |
QUGGVEQQEMGTDN
|
8.6 | IC50 | 2 | — | |
JXAAATVXBZVTFP
|
8.6 | IC50 | 2 | — | |
UZHHQLXSRNDLIY
|
8.6 | IC50 | 2 | — | |
MUSVRXWCIMGFPH
|
8.6 | IC50 | 2 | — | |
SCIQVOYRQAZVMN
|
8.5 | IC50 | 2 | — | |
QEEDOZCUASXVAK
|
8.5 | IC50 | 2 | — | |
QZFUHCFFTCONDW
|
8.4 | IC50 | 2 | — | |
CHLMMQSHPOCAPQ
|
8.3 | IC50 | 2 | — | |
XIPGMFZCORQMAY
|
8.3 | IC50 | 2 | — | |
MEICPLZXVLQHSW
|
8.3 | IC50 | 2 | — | |
JKHYOWBRQRJSTQ
|
8.2 | IC50 | 2 | — | |
KUYSMMDYWSPSDF
|
8.2 | IC50 | 2 | — | |
HVJUJYFSYHNRDU
|
8.2 | IC50 | 2 | — | |
ZPTKJYMGKHTPFV
|
8.1 | IC50 | 2 | — | |
OAOOUVFCVORAIE
|
8.1 | IC50 | 2 | — | |
HAQSIEIEPKZOHT
|
8.1 | IC50 | 2 | — | |
PMXMADULYZHDGE
|
8.1 | IC50 | 2 | — | |
MYJNLWYXNNVJAZ
|
8.0 | IC50 | 2 | — | |
PYHWTMOCTYEEAJ
|
7.9 | IC50 | 2 | — | |
GKJVTZJLHFEZJH
|
7.8 | IC50 | 2 | — | |
WGCXUGFPWKBWOP
|
7.8 | IC50 | 2 | — | |
SPCXYBUWDJJYRU
|
7.4 | IC50 | 2 | — | |
NGBACBJFDKYOER
|
7.4 | IC50 | 2 | — | |
KKNFPZSPEHSKQU
|
7.2 | IC50 | 2 | — | |
LDMOLCOFCNCFPU
|
6.9 | IC50 | 2 | — | |
TZNSZZMLARSGAI
|
6.9 | IC50 | 2 | — |