Target Details
| UniProt AC | P04085 |
|---|---|
| Gene Symbol | PDGFA |
| Protein Name | Platelet-derived growth factor subunit A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00341 (PDGF) PF04692 (PDGF_N) |
Summary
- Multi-target molecules 1
- Clinical molecules 0
- Avg pChEMBL 6.21
KEGG Pathways (20)
- Calcium signaling pathway
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Gap junction
- Glioma
- Integrin signaling
- JAK-STAT signaling pathway
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Associated Diseases (2)
Active Molecules (1)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OJFKUJDRGJSAQB
|
6.2 | IC50 | 17 | — |