Target Details
UniProt ACP04070
Gene SymbolPROC
Protein NameVitamin K-dependent protein C
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF14670 (FXa_inhibition) PF00594 (Gla) PF00089 (Trypsin)
Summary
  • Multi-target molecules 39
  • Clinical molecules 0
  • Avg pChEMBL 6.97
Top Co-occurrence Targets
Active Molecules (39)
InChIKey pChEMBL Type Targets Clinical
BHQDUYVBGREBCB 9.3 Ki 8
HJCCPKALMCCVEK 9.2 Ki 5
RCVRHAVSXLQPDX 9.2 Ki 5
AXXYATYQRMPQSN 8.7 Ki 6
DBLYNSSCIKMVDW 8.3 Ki 3
ZYKYKDNQGMXJQR 7.6 Ki 5
OXHLIVRHOPCUSV 7.4 Ki 5
UWAQLEGUXYPPDC 7.4 Ki 4
HLENBKTVSREWEE 7.4 Ki 8
UPFBONOEYAFXQG 7.3 Ki 5
ZTJVQQCXGUIYTL 7.2 Ki 4
RFKOYFYQZZFWKX 7.2 Ki 3
PDUMJXCNOKHQKH 7.1 Ki 9
MLPXCKVDBGAVRJ 7.1 Ki 3
XWJGZMVWOIPRDB 7.0 Ki 5
ONDHAMRPENUPCS 6.8 Ki 4
DEEHPLDVAKJVIC 6.8 IC50 2
FHJDRBBZAGYRKH 6.8 Ki 4
ZVYUEFHDJYEETD 6.7 Ki 5
BQJXMSPBOZFQJJ 6.7 Ki 4
WDJIHZCWTLEDHQ 6.7 IC50 2
YBLXUAHRYXEFCL 6.7 Ki 4
MLVTZWQEWUGCSC 6.7 Ki 5
DXGZDORACWBTJS 6.6 Ki 4
XSPHSWHLHARGRZ 6.6 IC50 2
OITRKHUOZGPBJI 6.5 Ki 4
AFGGMWNLRYRQDA 6.5 Ki 3
FDLUVBKZNIPEQR 6.4 Ki 6
IGCAUFKCIHSDQS 6.4 Ki 5
RATKUIDPANMWSA 6.3 Ki 2
MCDKKKIUEGNSPK 6.3 Ki 5
UIBUHBYTPNMHCK 6.2 Ki 5
JPGNXUNXIAMWMQ 6.2 Ki 5
VNKFZBCCJJVXJG 6.2 Ki 5
PROYMPSAMYSXNO 6.1 Ki 4
BJSIWIFJSRFHPS 6.1 Ki 6
YLOURKKYJRCESD 6.1 Ki 5
BVZHCUOVJATBQP 6.1 Ki 5
DOEPKHLCEFPBEX 6.1 Ki 4
2D structure