Target Details
| UniProt AC | P04062 |
|---|---|
| Gene Symbol | GBA1 |
| Protein Name | Lysosomal acid glucosylceramidase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02055 (Glyco_hydro_30) PF17189 (Glyco_hydro_30C) |
Summary
- Multi-target molecules 57
- Clinical molecules 0
- Avg pChEMBL 6.78
KEGG Pathways (5)
Associated Diseases (3)
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CEEPDUGFKXBMCP
|
8.5 | IC50 | 2 | — | |
MLRMIFDEZCZOAE
|
8.5 | IC50 | 2 | — | |
FETSBCRHESSCQO
|
8.3 | IC50 | 2 | — | |
GTFOIXYCSJUOKQ
|
8.3 | IC50 | 2 | — | |
JYUBGYMPVKAJEH
|
8.3 | IC50 | 2 | — | |
OMVDIWMZQBJVFN
|
8.3 | IC50 | 2 | — | |
KACLQPKKHWDLNL
|
8.1 | IC50 | 2 | — | |
UQDXIILZCYJPNV
|
7.7 | Ki | 2 | — | |
NJOZFAFEQVQFJI
|
7.6 | Ki | 2 | — | |
QPYJXFZUIJOGNX
|
7.5 | IC50 | 3 | — | |
TYXAKMAAZJJHCB
|
7.3 | IC50 | 2 | — | |
ZIOJXWDAAUVOFR
|
7.2 | IC50 | 2 | — | |
VZJFARCTRJANNN
|
7.2 | IC50 | 3 | — | |
UWQNTLVHUVARDK
|
7.0 | IC50 | 2 | — | |
JORKMVPNKKKNIS
|
7.0 | IC50 | 3 | — | |
BMDCVDRGQXCITF
|
6.9 | IC50 | 2 | — | |
XVYLNHVEAOOEGI
|
6.8 | IC50 | 5 | — | |
DWHQKLOFYPHDRY
|
6.7 | IC50 | 3 | — | |
HBNZOGWTAOYFRQ
|
6.7 | IC50 | 3 | — | |
IRIRASPSMMWZOM
|
6.7 | IC50 | 4 | — | |
PFYHYHZGDNWFIF
|
6.7 | Ki | 2 | — | |
XVYLNHVEAOOEGI
|
6.7 | IC50 | 4 | — | |
DWCDYYDNUCIAGD
|
6.6 | IC50 | 4 | — | |
GBGOUGJOHMBDPJ
|
6.6 | IC50 | 3 | — | |
GMGNEDCNRHODKX
|
6.6 | IC50 | 3 | — | |
VYGIZBXHTDCYFB
|
6.6 | IC50 | 3 | — | |
YMWWYTOTURKGDE
|
6.6 | IC50 | 3 | — | |
DKPSDLOOZAIQNL
|
6.5 | IC50 | 4 | — | |
FTSCEGKYKXESFF
|
6.5 | IC50 | 2 | — | |
JLJXOROVAFNSCP
|
6.5 | IC50 | 3 | — | |
JWYVFZRNNGAAIG
|
6.5 | IC50 | 4 | — | |
MGIKPOPLRLHKKL
|
6.5 | IC50 | 4 | — | |
CHMJMOCFEUVONE
|
6.5 | IC50 | 3 | — | |
ISWDTKRAKJESLP
|
6.5 | IC50 | 2 | — | |
IIHXPVAHXKBRBL
|
6.4 | IC50 | 2 | — | |
BXIWEAVNUFIVND
|
6.4 | IC50 | 3 | — | |
IYBACZJBAZUVGN
|
6.4 | IC50 | 4 | — | |
PGOGHEZNHFQKSP
|
6.4 | IC50 | 3 | — | |
NCWNCLLUJRRPFV
|
6.4 | IC50 | 2 | — | |
CJZGTRIZBSILBI
|
6.3 | IC50 | 3 | — | |
IMYBJLKJUZUZCD
|
6.3 | IC50 | 3 | — | |
NGXJLNWOFGXCDY
|
6.3 | IC50 | 2 | — | |
RONFUEZMVTVAJF
|
6.3 | IC50 | 3 | — | |
SXPLUAKSZJTQBC
|
6.3 | IC50 | 2 | — | |
WHMRDWKWVDYZNI
|
6.3 | IC50 | 3 | — | |
XWORIPUWULNBFL
|
6.3 | IC50 | 3 | — | |
ZDHLSZPFRBINKG
|
6.3 | IC50 | 2 | — | |
UREJDUPKGMFJRU
|
6.2 | IC50 | 17 | — | |
VGSQNAQYXKTCLP
|
6.2 | IC50 | 2 | — | |
UPTPKEASQZRVIR
|
6.2 | IC50 | 3 | — |