Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGCHRDUVHNVKAK
|
7.7 | IC50 | 2 | Yes | |
KGUVBHLPMGERAT
|
7.7 | IC50 | 8 | Yes | |
LPZWIAVKYXCHGC
|
7.7 | IC50 | 7 | Yes | |
MGQZHWBYKGXMDX
|
7.7 | IC50 | 5 | Yes | |
NWVCPUQBLORAAX
|
7.7 | IC50 | 3 | — | |
VLTOUUSTKONGKC
|
7.7 | Ki | 10 | Yes | |
WBTHKLMTSOWADI
|
7.7 | IC50 | 2 | — | |
WICQDDCNCVTFDX
|
7.7 | Ki | 16 | Yes | |
XNLVNQQMTWGGIM
|
7.7 | IC50 | 5 | Yes | |
YBQLENDMILTZBB
|
7.7 | IC50 | 6 | Yes | |
YIYXDKFJIKECAM
|
7.7 | IC50 | 5 | Yes | |
AOPSFGSGYVNAEJ
|
7.7 | IC50 | 5 | Yes | |
BDRKJDRHTIDJDK
|
7.7 | IC50 | 5 | Yes | |
BPNDGQNQHSBNOE
|
7.7 | IC50 | 7 | Yes | |
HTNLSTWGHBHDPS
|
7.7 | IC50 | 8 | Yes | |
JYIVEWZWGSXEIG
|
7.7 | Ki | 5 | Yes | |
QRDYOYPORKWZCP
|
7.7 | IC50 | 6 | Yes | |
QYFKTMNLZHLRIH
|
7.7 | IC50 | 7 | Yes | |
SUSMVCKSLVPRCL
|
7.7 | IC50 | 7 | Yes | |
UVBJVUYVRZYYHC
|
7.7 | IC50 | 5 | Yes | |
DFPDFXUEOXPMIV
|
7.7 | Ki | 7 | Yes | |
SUSMVCKSLVPRCL
|
7.7 | IC50 | 5 | — | |
COUUBDFXGTZTPW
|
7.6 | Ki | 5 | Yes | |
WFVYENBQHIIIQE
|
7.6 | IC50 | 7 | Yes | |
ACSSJLXQNWFMSO
|
7.6 | Ki | 7 | Yes | |
CBMKHOZXSARYNG
|
7.6 | IC50 | 6 | Yes | |
DNGGPLKVDUPXFN
|
7.6 | IC50 | 5 | — | |
DNGGPLKVDUPXFN
|
7.6 | IC50 | 7 | Yes | |
FAEZTVRCESNVJN
|
7.6 | IC50 | 6 | Yes | |
FMPSZEWYBZCYDN
|
7.6 | IC50 | 6 | Yes | |
FXAWYNXKIRKVPJ
|
7.6 | IC50 | 3 | Yes | |
JGJZJJQMNAKKDG
|
7.6 | Ki | 7 | Yes | |
LMASIGSKSCEZDY
|
7.6 | IC50 | 5 | Yes | |
MCSWSPNUKWMZHM
|
7.6 | IC50 | 7 | Yes | |
PIHNCDLSZQOOPU
|
7.6 | Ki | 6 | Yes | |
UTERPWJSMDDIGY
|
7.6 | Ki | 8 | Yes | |
YBRVBUDXSMPLGQ
|
7.6 | IC50 | 5 | Yes | |
AKWKBACKRMYPRV
|
7.6 | Ki | 6 | Yes | |
AWBXCXPCFJCVSM
|
7.6 | IC50 | 4 | — | |
CNZGQRARNYMASL
|
7.6 | Ki | 7 | Yes | |
FAFCWIZUCJNALJ
|
7.6 | IC50 | 2 | — | |
GHHVNOZFZMDYFQ
|
7.6 | Ki | 7 | Yes | |
GTXSRFUZSLTDFX
|
7.6 | IC50 | 5 | — | |
GTXSRFUZSLTDFX
|
7.6 | IC50 | 8 | Yes | |
HLJHTDAQDAFOFS
|
7.6 | Ki | 7 | Yes | |
IHPUTEIJIZVYPC
|
7.6 | Ki | 7 | Yes | |
INSQINPAEQOIQL
|
7.6 | IC50 | 7 | Yes | |
NEUXHEKNAOUEQU
|
7.6 | Ki | 7 | Yes | |
PKGJPJPGFGLRRN
|
7.6 | IC50 | 2 | — | |
SSQXFNKOLMHXPO
|
7.6 | Ki | 6 | Yes |