Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DPQCHTZYBRQXQC
|
8.0 | Ki | 7 | Yes | |
NQUUIXIBNFFYTG
|
8.0 | Ki | 6 | Yes | |
CHAFUQVXOKHDCA
|
8.0 | Ki | 5 | Yes | |
FITSVZFOIGFQQI
|
8.0 | Ki | 6 | Yes | |
IWQSGINKBSWILJ
|
8.0 | IC50 | 10 | — | |
LNSULHYVZXTWFG
|
8.0 | Ki | 4 | Yes | |
LWZOHIDILGLXGF
|
8.0 | IC50 | 5 | Yes | |
SPVUAASKZWLIQS
|
8.0 | IC50 | 5 | Yes | |
UOLDAWOAHWACHY
|
8.0 | IC50 | 3 | — | |
USDAGEMRRVCVKK
|
8.0 | IC50 | 3 | Yes | |
JMWYGNIQHYKDCH
|
8.0 | Ki | 7 | Yes | |
MXGYLPKHTGTZKG
|
7.9 | Ki | 7 | Yes | |
MZISFPSOTJFTTJ
|
7.9 | Ki | 7 | Yes | |
HGYBTJHBZBLHNW
|
7.9 | IC50 | 3 | Yes | |
LDNXMPSGDXDZPD
|
7.9 | IC50 | 3 | Yes | |
SESYXDSEOCRODR
|
7.9 | Ki | 7 | Yes | |
ATNNMKHWMHMLHP
|
7.9 | Ki | 7 | Yes | |
BEKYMPWGANBKBK
|
7.9 | Ki | 7 | Yes | |
DONMTDNLNMLOIC
|
7.9 | Ki | 13 | Yes | |
JQYSJWITJMOASO
|
7.9 | IC50 | 6 | Yes | |
NVNGYUBMJMOHQL
|
7.9 | IC50 | 6 | Yes | |
QHCDOFQMQJCFGF
|
7.9 | IC50 | 4 | — | |
RCJJPUINEATAJF
|
7.9 | Ki | 4 | Yes | |
RRETZYBLLSHELY
|
7.9 | IC50 | 6 | Yes | |
ZJYCLDORACELQK
|
7.9 | Ki | 3 | — | |
GETQXLAMYOMSJS
|
7.9 | IC50 | 8 | Yes | |
MMCVYPKEJGVLMH
|
7.9 | Ki | 7 | Yes | |
BJBDOOZTEPGOJP
|
7.8 | IC50 | 5 | Yes | |
BLCLPMFYNMXITO
|
7.8 | IC50 | 5 | Yes | |
HXFIFSALSXGAFS
|
7.8 | Ki | 4 | Yes | |
RHOVUJYSXPHHFW
|
7.8 | IC50 | 2 | — | |
RVZWFNDDFJIWNJ
|
7.8 | IC50 | 2 | — | |
YLXVWRCBKXEQFD
|
7.8 | IC50 | 6 | Yes | |
WPXAJFJACNOICK
|
7.8 | Ki | 7 | Yes | |
BEWFNUZAYXMBNS
|
7.8 | IC50 | 5 | Yes | |
CYBDDZKSRZPTQR
|
7.8 | IC50 | 6 | Yes | |
DCSHLVVGHNRVCO
|
7.8 | Ki | 7 | Yes | |
FRRDNYNCIZOSSI
|
7.8 | IC50 | 5 | Yes | |
GTBJTISRJIZWKE
|
7.8 | IC50 | 7 | Yes | |
OHYRHJPFKZKXOS
|
7.8 | Ki | 4 | Yes | |
RSMQCSLXBNSQJJ
|
7.8 | Ki | 7 | Yes | |
VURZBHKGMIEEFK
|
7.8 | Ki | 7 | Yes | |
KOFNJKLYWDTWHZ
|
7.8 | Ki | 7 | Yes | |
RCGPSTRFXVIUQB
|
7.8 | Ki | 7 | Yes | |
BGNATPVKWHRROW
|
7.8 | Ki | 6 | Yes | |
CDVYEYANHXGLCX
|
7.8 | Ki | 10 | Yes | |
DIIAIQCOHXBJHI
|
7.8 | IC50 | 6 | Yes | |
DXDRHHKMWQZJHT
|
7.8 | IC50 | 9 | — | |
PECNGMJVFOGIBW
|
7.8 | IC50 | 7 | Yes | |
PJKBQUWSOBIDMI
|
7.8 | Ki | 4 | Yes |