Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXXIQAWIZFAIOP
|
8.2 | Ki | 9 | Yes | |
CVZIHNYAZLXRRS
|
8.2 | IC50 | 10 | Yes | |
CVZIHNYAZLXRRS
|
8.2 | IC50 | 6 | Yes | |
GFUITADOEPNRML
|
8.2 | IC50 | 8 | Yes | |
HNXQLWUITFQYPE
|
8.2 | Ki | 10 | Yes | |
MOPRTFSMCQNUCT
|
8.2 | IC50 | 9 | Yes | |
QVXRAVFETVTALN
|
8.2 | IC50 | 5 | Yes | |
SHTYCRVVDNRZDY
|
8.2 | IC50 | 5 | Yes | |
SNYKGOMEURTYMK
|
8.2 | Ki | 10 | Yes | |
XFNJKSWXHKYCFN
|
8.2 | Ki | 10 | Yes | |
ZYZUZMRFPDIWGW
|
8.2 | IC50 | 5 | Yes | |
PCAPSCAFNCUGDE
|
8.1 | Ki | 6 | Yes | |
ABTPKZSVAHUDFA
|
8.1 | Ki | 5 | Yes | |
GSWRTFGMHRKLKT
|
8.1 | IC50 | 14 | Yes | |
JFMSSTVXWKCAJH
|
8.1 | Ki | 7 | Yes | |
ABOVSYRJLZIGMD
|
8.1 | Ki | 5 | Yes | |
IQTIGUJOCAYBRM
|
8.1 | IC50 | 3 | Yes | |
RYRSPABEKSPRKC
|
8.1 | IC50 | 7 | Yes | |
VWEKUHYRCOZNGA
|
8.1 | IC50 | 2 | — | |
WLWNRAWQDZRXMB
|
8.1 | Ki | 6 | Yes | |
MQLHBSAEUUVJRX
|
8.1 | IC50 | 6 | Yes | |
YKPYIPVDTNNYCN
|
8.1 | IC50 | 11 | Yes | |
YUWSFQQPCKKPJG
|
8.1 | IC50 | 9 | Yes | |
WIUDGBCTJVXBCM
|
8.1 | IC50 | 7 | — | |
LDMWZYZAAZFUTC
|
8.1 | IC50 | 2 | — | |
GKHRDWHFKKUYAX
|
8.1 | IC50 | 9 | — | |
JBVXKMHBLNDBBV
|
8.1 | IC50 | 6 | Yes | |
LRVIJTRFTUQDKW
|
8.1 | IC50 | 7 | Yes | |
LXSYXSGOVAASBA
|
8.1 | IC50 | 6 | Yes | |
OKYUILRERWOFCH
|
8.1 | IC50 | 7 | Yes | |
TUXGRLPRNXNACO
|
8.1 | IC50 | 5 | Yes | |
UERCGTJUVRFNRO
|
8.1 | Ki | 6 | Yes | |
VYGKNAIULXUTGK
|
8.0 | IC50 | 6 | Yes | |
FOCKEUBBGLJYBX
|
8.0 | IC50 | 5 | Yes | |
PTSHMCCZVCAMNJ
|
8.0 | Ki | 6 | Yes | |
AALOSJKQIIRSAO
|
8.0 | IC50 | 6 | Yes | |
GWEITLSXCOXESW
|
8.0 | IC50 | 7 | Yes | |
IRBWGGQXMBAYQL
|
8.0 | IC50 | 7 | Yes | |
LRYRCUJGWNCKPO
|
8.0 | IC50 | 5 | Yes | |
QHRUJPVXLYJUEM
|
8.0 | IC50 | 6 | Yes | |
REPZHAUIJREHGP
|
8.0 | Ki | 3 | Yes | |
RYMINZKMUZXTLF
|
8.0 | IC50 | 6 | Yes | |
VDDKIBQLKXMKIW
|
8.0 | Ki | 7 | Yes | |
WJPFHUMULGZBAI
|
8.0 | IC50 | 4 | Yes | |
WORSVFBVUCBRIP
|
8.0 | IC50 | 5 | — | |
XGFRXSAFARHCLC
|
8.0 | IC50 | 5 | Yes | |
XNKSQYFVFJZMOA
|
8.0 | IC50 | 7 | Yes | |
ZWDYAHGBOJEURS
|
8.0 | IC50 | 5 | Yes | |
KFUADVZPCULIED
|
8.0 | Ki | 7 | Yes | |
ZJYCLDORACELQK
|
8.0 | Ki | 5 | Yes |