Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AIBDPCDNFOFGFS
|
8.3 | Ki | 6 | Yes | |
RBLCSCFFNCADJO
|
8.3 | Ki | 5 | — | |
RBLCSCFFNCADJO
|
8.3 | Ki | 7 | Yes | |
RBLCSCFFNCADJO
|
8.3 | Ki | 5 | — | |
XEONYLBJVDXPRB
|
8.3 | IC50 | 6 | Yes | |
SGQBRJNZCHCINW
|
8.3 | IC50 | 6 | Yes | |
QQWABDFFKSDQLH
|
8.3 | IC50 | 6 | Yes | |
QRXOZHSEEGNRFC
|
8.3 | IC50 | 8 | Yes | |
USYXNFCQBGQYRW
|
8.3 | Ki | 6 | Yes | |
FEWWJFPIJXNCFE
|
8.3 | Ki | 7 | Yes | |
IOTJDDOXTYOJJN
|
8.3 | IC50 | 6 | Yes | |
OCSMOTCMPXTDND
|
8.3 | IC50 | 8 | Yes | |
OEPLGUBYTRYCJX
|
8.3 | IC50 | 7 | Yes | |
PNKICJSNJYXQOE
|
8.3 | IC50 | 3 | — | |
QRXOZHSEEGNRFC
|
8.3 | IC50 | 8 | Yes | |
UDNLRUDZHBXCON
|
8.3 | Ki | 7 | Yes | |
ZAXDLNVDZOYNCA
|
8.3 | IC50 | 6 | Yes | |
ZBTKKYFIZQHNDQ
|
8.3 | IC50 | 7 | Yes | |
DZVQTAQHEPKNSI
|
8.3 | IC50 | 6 | Yes | |
MAOGHLYYLNCNCI
|
8.3 | IC50 | 7 | Yes | |
CFUYAVWBVRZFLA
|
8.3 | Ki | 6 | Yes | |
WLWNRAWQDZRXMB
|
8.3 | Ki | 6 | Yes | |
LICJLIVFDQFASY
|
8.3 | Ki | 6 | Yes | |
YOZKFIDLBXLPFF
|
8.3 | IC50 | 7 | Yes | |
GAQJSKIBXSLAJK
|
8.2 | IC50 | 6 | Yes | |
YTRMRJDVKQXSIU
|
8.2 | IC50 | 4 | Yes | |
FCGVXISUYVDDPU
|
8.2 | IC50 | 7 | Yes | |
HOGIHVAAHRAULF
|
8.2 | IC50 | 5 | Yes | |
IXEFVZDHNHSUSD
|
8.2 | IC50 | 5 | Yes | |
MVRHXCGLUWVMKH
|
8.2 | IC50 | 7 | Yes | |
OHZMUNMVWGUMMY
|
8.2 | IC50 | 6 | Yes | |
QKOVHOITGZCHQW
|
8.2 | IC50 | 4 | Yes | |
QYZPDCGWIJYZMN
|
8.2 | IC50 | 8 | Yes | |
RAPHEYPJGISJNU
|
8.2 | Ki | 10 | Yes | |
ROMGJVVZNVJOPW
|
8.2 | Ki | 10 | Yes | |
XMUJRKRMNALZLF
|
8.2 | IC50 | 2 | — | |
YLYMDJMYRSEUOA
|
8.2 | IC50 | 7 | Yes | |
YYRRVFYCIQQYHU
|
8.2 | Ki | 6 | Yes | |
YZDALJROFHNCEI
|
8.2 | IC50 | 3 | Yes | |
ZVAKMIZOMSWYGQ
|
8.2 | IC50 | 7 | Yes | |
LXWSFODDORIHFJ
|
8.2 | IC50 | 6 | Yes | |
SLHHOJZYTMNFRR
|
8.2 | Ki | 6 | Yes | |
YKYLOHCKSMYHPL
|
8.2 | IC50 | 6 | Yes | |
DZWVTHAIOWIVNT
|
8.2 | Ki | 7 | Yes | |
HEPINVNDBLHRTM
|
8.2 | IC50 | 6 | Yes | |
KMYAHTGTYRRWEK
|
8.2 | Ki | 6 | Yes | |
GMNFREWQYNXZAF
|
8.2 | Ki | 7 | Yes | |
HFKQCTSECBMUHK
|
8.2 | IC50 | 4 | Yes | |
CEEASCNCHQSPKF
|
8.2 | IC50 | 5 | Yes | |
NWIDFBAHFQXVFF
|
8.2 | IC50 | 5 | Yes |