Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LBZOGBFXCHOCBC
|
8.7 | IC50 | 6 | Yes | |
BKTXYTRQOBRSNS
|
8.7 | IC50 | 2 | — | |
FTWOUUKMIDBQOJ
|
8.7 | IC50 | 2 | — | |
GKHRDWHFKKUYAX
|
8.7 | IC50 | 8 | Yes | |
MHQJDNZHPIZRRV
|
8.7 | IC50 | 4 | — | |
SLHHOJZYTMNFRR
|
8.7 | Ki | 7 | Yes | |
VCJOCQOXJUMEBE
|
8.7 | IC50 | 6 | Yes | |
GFUITADOEPNRML
|
8.6 | Ki | 11 | Yes | |
KOLIYILUYWKKNC
|
8.6 | Ki | 4 | Yes | |
NMAKKNGSMZZSBP
|
8.6 | IC50 | 4 | Yes | |
PZPOCZWOYXDPDG
|
8.6 | IC50 | 5 | Yes | |
YKHOQKKUOWOUDP
|
8.6 | Ki | 2 | — | |
SCRXVDGCFAHYTL
|
8.6 | IC50 | 2 | — | |
TVNINFNNQVBJHI
|
8.6 | IC50 | 8 | Yes | |
WMYJDFANEQLDGP
|
8.6 | IC50 | 6 | — | |
DNFCKYUQJJTPGW
|
8.6 | IC50 | 2 | — | |
JMYNELQJPYBCPZ
|
8.6 | IC50 | 6 | Yes | |
WWNOVCQMRIZSRV
|
8.6 | IC50 | 8 | Yes | |
BZTWELLPCHJZLB
|
8.6 | IC50 | 6 | Yes | |
LFRIKIYAMSRRPD
|
8.6 | IC50 | 5 | Yes | |
QPPXLNJKZJGLRN
|
8.6 | IC50 | 6 | Yes | |
PGWQPFWCLKSUIC
|
8.6 | Ki | 5 | Yes | |
YAWCEEHWRJZVNM
|
8.6 | IC50 | 2 | — | |
MMRISAVXAFHOJP
|
8.5 | IC50 | 4 | Yes | |
RHWGGEKVTPKRQW
|
8.5 | IC50 | 4 | Yes | |
VCUJZXCWHYPIIH
|
8.5 | IC50 | 5 | Yes | |
AKNDZTHCJLFZCF
|
8.5 | IC50 | 9 | Yes | |
AKPXMDCVGKJBIP
|
8.5 | Ki | 4 | Yes | |
ANFAAJVPGXQKBB
|
8.5 | IC50 | 6 | Yes | |
FPSMXPGSVWPWCG
|
8.5 | IC50 | 8 | — | |
GFUITADOEPNRML
|
8.5 | Ki | 6 | — | |
GWQRQVFEMGHPMD
|
8.5 | Ki | 10 | Yes | |
HFAGTNGCAZYYLZ
|
8.5 | Ki | 13 | Yes | |
JCVSSJUXUIJGBT
|
8.5 | IC50 | 5 | Yes | |
KXEGEKRSCUZQMH
|
8.5 | IC50 | 5 | Yes | |
OFCWIPGKPUJTDP
|
8.5 | IC50 | 7 | Yes | |
OONXADPQRATYFL
|
8.5 | Ki | 5 | Yes | |
USIBDKCJHKIPNX
|
8.5 | IC50 | 6 | Yes | |
MVNUXJNXEWKALY
|
8.5 | IC50 | 5 | Yes | |
TZNUGSCRBFBAFR
|
8.5 | Ki | 7 | Yes | |
DYKLASPWVUKEIT
|
8.5 | IC50 | 6 | Yes | |
GKLAUAGSCYZMQP
|
8.5 | Ki | 7 | Yes | |
RTKNMWBYPISZDZ
|
8.4 | Ki | 7 | Yes | |
YJNJISQXBXDEOV
|
8.4 | IC50 | 4 | Yes | |
DJASZHFLBWUJAJ
|
8.4 | Ki | 7 | Yes | |
MTDVSXPXWCWOED
|
8.4 | IC50 | 6 | Yes | |
QXLMMZHXXOWCDY
|
8.4 | IC50 | 4 | Yes | |
WBONEAZKRBRCNC
|
8.4 | Ki | 4 | Yes | |
CDUNTBSHRUTDFM
|
8.4 | Ki | 7 | Yes | |
FQRZOEBSTPAQBJ
|
8.4 | IC50 | 4 | — |