Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SWRNCXLTVBBIMK
|
7.4 | IC50 | 7 | Yes | |
TVRLHUWRJSTBAB
|
7.4 | IC50 | 6 | Yes | |
WYVILPRSBDCCKY
|
7.4 | Ki | 7 | Yes | |
XJMLKUIRAXOATH
|
7.4 | IC50 | 7 | Yes | |
XVUIGVGFVWRFJO
|
7.4 | Ki | 4 | — | |
XVUIGVGFVWRFJO
|
7.4 | IC50 | 8 | Yes | |
ALZQLPXUMAEFBO
|
7.4 | IC50 | 3 | Yes | |
ATFPFLNWBZIBTJ
|
7.4 | IC50 | 6 | Yes | |
IBUXWZOBVVWCHD
|
7.4 | Ki | 7 | Yes | |
IPBVPRHDESNKFG
|
7.4 | Ki | 6 | Yes | |
JZKQUJKQSKTEON
|
7.4 | IC50 | 6 | Yes | |
YLQBSSFZOXXRNR
|
7.4 | IC50 | 6 | Yes | |
YZOKWMYHTLQIDP
|
7.4 | IC50 | 5 | Yes | |
GDBNAEMVDGQOCE
|
7.4 | IC50 | 7 | — | |
JMLWJDXZFPKMED
|
7.4 | IC50 | 2 | Yes | |
JVBPIOHSXSYBRG
|
7.4 | Ki | 7 | Yes | |
UWHDYIJAXRNLQS
|
7.4 | Ki | 6 | Yes | |
YVJXBWDNNWDVMN
|
7.4 | IC50 | 9 | Yes | |
ZPYLLHLHJRMHKM
|
7.4 | IC50 | 4 | Yes | |
IQHWFMFCBUDMAF
|
7.4 | Ki | 6 | Yes | |
TZYCKWCFYXFTIR
|
7.4 | IC50 | 5 | Yes | |
WIWASQOQNPNFMY
|
7.4 | IC50 | 5 | Yes | |
XGJAXXYDMLECBQ
|
7.4 | IC50 | 7 | Yes | |
ZCJSXQVUNXJVQQ
|
7.4 | IC50 | 2 | — | |
KXZZWRQJKQVMKR
|
7.4 | IC50 | 7 | Yes | |
ZGSTVUAZFACDLH
|
7.4 | IC50 | 4 | — | |
ZGSTVUAZFACDLH
|
7.4 | Ki | 8 | Yes | |
BYBOLCACCXBYNF
|
7.4 | IC50 | 4 | Yes | |
OVKVSVACJPYFHM
|
7.4 | IC50 | 5 | Yes | |
VKUYLANQOAKALN
|
7.4 | Ki | 7 | Yes | |
DRXVUBODYFAEED
|
7.3 | IC50 | 4 | — | |
IHXYDMMVEDLUPK
|
7.3 | IC50 | 3 | Yes | |
KPJZJSWNHXZALM
|
7.3 | IC50 | 5 | Yes | |
OPYOHFRGHGDNSJ
|
7.3 | Ki | 7 | Yes | |
UOLDAWOAHWACHY
|
7.3 | IC50 | 2 | — | |
ZORDGSDKVXISJV
|
7.3 | IC50 | 6 | Yes | |
CVMOEYXHQALNTG
|
7.3 | Ki | 6 | Yes | |
FUXYTSOUUZCQPA
|
7.3 | IC50 | 7 | — | |
JRUBYRGXZQLBRV
|
7.3 | IC50 | 2 | — | |
NTWPNMLRTBRVIB
|
7.3 | IC50 | 5 | Yes | |
VILDLUTXDBUVFM
|
7.3 | IC50 | 2 | Yes | |
FKPCCEUCLYUJQA
|
7.3 | IC50 | 6 | Yes | |
HXAROWWJPCDNRW
|
7.3 | IC50 | 6 | Yes | |
MOBAWCSMNMHMJW
|
7.3 | IC50 | 4 | Yes | |
UGEYJONPMBOKNN
|
7.3 | IC50 | 7 | Yes | |
UQRFKNRXERPSMG
|
7.3 | IC50 | 5 | Yes | |
XRAGTWOVABKXJS
|
7.3 | IC50 | 4 | Yes | |
NQPIHEUUYRAYII
|
7.3 | IC50 | 8 | Yes | |
RMDCZACTUKUROI
|
7.3 | IC50 | 5 | Yes | |
SSVAOOCBANMUMS
|
7.3 | IC50 | 5 | Yes |