Target Details
| UniProt AC | P03956 |
|---|---|
| Gene Symbol | MMP1 |
| Protein Name | Interstitial collagenase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,338
- Clinical molecules 1178
- Avg pChEMBL 7.11
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GCBPAPVOMPJQHK
|
10.0 | Ki | 9 | Yes | |
QVHQLFLTQMCYLJ
|
9.6 | IC50 | 6 | Yes | |
OBJBBLBMOOBABD
|
9.5 | IC50 | 8 | Yes | |
ULILDPSFFUSXJH
|
9.4 | IC50 | 9 | Yes | |
ULILDPSFFUSXJH
|
9.4 | IC50 | 7 | — | |
KYOFVPKPPTUVKK
|
9.3 | IC50 | 8 | Yes | |
YTCCTPYUECNUFO
|
9.3 | IC50 | 7 | Yes | |
MOODLLAARDEUNJ
|
9.2 | Ki | 6 | Yes | |
SRVJEHMEZKLIMK
|
9.2 | Ki | 4 | Yes | |
MWYSQPGMUZLIHV
|
9.2 | Ki | 6 | Yes | |
NRCQPJPKKZDRND
|
9.2 | Ki | 6 | Yes | |
XSWDEIOVOAQSMZ
|
9.2 | IC50 | 7 | Yes | |
CYYCSKFJEOSZTF
|
9.1 | IC50 | 9 | Yes | |
JTCBZWXCQOLSNN
|
9.1 | IC50 | 2 | — | |
XDJHCLNLKWGZCM
|
9.1 | Ki | 5 | Yes | |
NQYWUYPYYFALAI
|
9.0 | Ki | 6 | Yes | |
IZYWROOEWSDARX
|
9.0 | Ki | 6 | Yes | |
KLSLMSQYLRDFGN
|
9.0 | IC50 | 5 | Yes | |
NEGPFWDWNNSJRQ
|
9.0 | Ki | 2 | — | |
OLEYZXUQGOKVKT
|
9.0 | IC50 | 7 | Yes | |
TUSYEXLVYIINDP
|
9.0 | IC50 | 6 | Yes | |
XFILPEOLDIKJHX
|
9.0 | IC50 | 12 | Yes | |
XXOLBMKULOJKQR
|
9.0 | IC50 | 7 | Yes | |
IOLRUMINDIUCLJ
|
9.0 | Ki | 8 | Yes | |
DDRBOOUOUSFWET
|
9.0 | IC50 | 4 | — | |
MDENDLKFAFTBOF
|
9.0 | IC50 | 2 | — | |
PJKWYBIJVPNFJI
|
9.0 | IC50 | 6 | Yes | |
AAPPTEGQHHRRCP
|
8.9 | IC50 | 6 | Yes | |
JIZLXLHASQJXJD
|
8.9 | IC50 | 2 | — | |
QPEZTCMCOIDQRV
|
8.9 | IC50 | 5 | Yes | |
RMKNDVDQYWXAON
|
8.9 | IC50 | 7 | Yes | |
USEJKZYMWYHGSP
|
8.9 | Ki | 7 | Yes | |
GPENKXZRTRUYOG
|
8.9 | IC50 | 4 | Yes | |
JBRUCLKAHIYELE
|
8.9 | IC50 | 3 | — | |
IKFMCZJWBBXODH
|
8.8 | Ki | 3 | Yes | |
OCSMOTCMPXTDND
|
8.8 | IC50 | 14 | Yes | |
RMMUGCXFUHIPQO
|
8.8 | IC50 | 2 | — | |
DJQJEICJRBFEOV
|
8.8 | IC50 | 4 | Yes | |
BJOZETKUSDMMAN
|
8.7 | IC50 | 6 | Yes | |
LKMAUWKMMZAHHV
|
8.7 | Ki | 5 | Yes | |
QSFJZGINKPYVRC
|
8.7 | Ki | 7 | Yes | |
AHBFOOOWLVWQFO
|
8.7 | IC50 | 6 | Yes | |
CQRAUIRVDKNRIO
|
8.7 | IC50 | 9 | Yes | |
FXEYKJYOHRTUNG
|
8.7 | IC50 | 6 | Yes | |
ZHLANTZRDCBWFM
|
8.7 | IC50 | 6 | Yes | |
JBYQQXSCANNDNP
|
8.7 | Ki | 4 | Yes | |
KNCYWVRUUBOHGE
|
8.7 | Ki | 7 | Yes | |
NITYDPDXAAFEIT
|
8.7 | IC50 | 20 | Yes | |
ZRDGYJAMDSHROJ
|
8.7 | IC50 | 7 | Yes | |
ZWHGUGYVAMXPJZ
|
8.7 | IC50 | 5 | Yes |