Target Details
UniProt ACP03952
Gene SymbolKLKB1
Protein NamePlasma kallikrein
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00024 (PAN_1) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,277
  • Clinical molecules 0
  • Avg pChEMBL 7.55
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,277)
InChIKey pChEMBL Type Targets Clinical
FZRJFARUZQXZOZ 8.1 IC50 2
QKFCYPKTTJCUSZ 8.1 Ki 8
XCPKGBCGNUMCNT 8.1 IC50 2
LCMPWMFTZAUSIJ 8.1 IC50 3
QEUZUPMZRYSKJR 8.1 IC50 2
XPUMGIIZTYUOQT 8.1 IC50 2
DEZNHCICTWBFEH 8.1 Ki 2
KXSZMPGKDDBJRE 8.1 IC50 3
QGNJMTPKSKWTBQ 8.1 IC50 2
XTUFVXUJJQAYGD 8.1 Ki 3
ZLYCPBBJASZKFG 8.1 Ki 4
ZWZWZPJQIZBWFH 8.1 IC50 2
ZYKYKDNQGMXJQR 8.1 Ki 5
HRLKIYSEPAYSAH 8.0 Ki 2
METWKYXLYOAEDA 8.0 IC50 2
GNLXHDHFJKLSJD 8.0 IC50 2
JPGNXUNXIAMWMQ 8.0 Ki 5
XWJGZMVWOIPRDB 8.0 Ki 4
XWJGZMVWOIPRDB 8.0 Ki 5
DDOFNAVOJKWETH 8.0 IC50 2
DJUCOOVKTPLJLE 8.0 Ki 2
FPAKZDLGEHHCTC 8.0 IC50 2
LNKXXEMOPNVZGM 8.0 Ki 2
XQGAAZGSIZFZJH 8.0 IC50 2
ZZXQOEFXCPENDW 8.0 IC50 2
KQZYQOJQXJGZMI 8.0 IC50 2
RLFXIFOZOPMNCY 8.0 IC50 2
AGDBQILBKXGVMA 8.0 IC50 2
ASWFFXNYMLHVMO 8.0 Ki 2
FJMCAFXMYKYZAO 8.0 Ki 3
GGKPWIXGKBVTFC 8.0 Ki 2
NVKNABMCMNHCSO 8.0 Ki 3
NWAGTUQRZPXSNY 8.0 IC50 5
OVHZQHDFJHZRDI 8.0 IC50 2
PBXKTYJYARTPQU 8.0 IC50 2
PODBMIDYMFKRKE 8.0 Ki 2
RTIMPDQMXMBUMW 8.0 IC50 2
SITZZDVPGOZBMP 8.0 Ki 3
SVNKORJSWJTHRX 8.0 IC50 2
SVTFEVREYQHXOM 8.0 IC50 2
XOPHHKQWDWBCDG 8.0 IC50 5
LPSATGNYPUSCRA 8.0 Ki 2
RKJMKFUCSWGOSU 8.0 Ki 2
DYNSAJCVHKUDFF 8.0 IC50 2
LUIFJTITJHESQD 8.0 Ki 2
CVGKJPRJDXNZKV 8.0 IC50 2
DCFGHORVDDAJPY 8.0 IC50 2
DERODARCDQXYDI 8.0 IC50 2
NAFNAAZYCZFUNR 8.0 IC50 2
NAVJAUKFYAXRGE 8.0 IC50 2
2D structure