Target Details
UniProt ACP03952
Gene SymbolKLKB1
Protein NamePlasma kallikrein
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00024 (PAN_1) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,277
  • Clinical molecules 0
  • Avg pChEMBL 7.55
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,277)
InChIKey pChEMBL Type Targets Clinical
LLJXUBIQRITYHZ 8.2 Ki 2
MWSHJNLPNRIIFT 8.2 Ki 3
OUALKAWDVQPBGH 8.2 IC50 2
WCANIIANZRELQI 8.2 IC50 2
YZJXJVFIOXDWAC 8.2 Ki 2
NHTJCIPCROASOS 8.2 IC50 2
KHTRQHPDTKFMGV 8.2 IC50 3
REWLFHBRHNXKCO 8.2 Ki 2
ROMIPLLXTVGFPF 8.2 IC50 2
XWNDSMYHTNPVSM 8.2 Ki 2
GTMQLRVEOBBFGO 8.2 Ki 3
QFMWDGOSYMZTRR 8.2 IC50 2
VABZDZOISVDIRI 8.2 Ki 3
NKCIMLZZOJBOGZ 8.2 IC50 2
SSZTYGHNKCZYAF 8.2 IC50 2
SYZUSCSRAOJBQO 8.2 IC50 2
QCAYWCRUVAGYIH 8.2 IC50 2
XMGACJAVDNSYFS 8.2 IC50 2
QGEHSULTCOSTKP 8.2 Ki 3
SNUMNATTXKTJQD 8.2 IC50 2
XAYFQGTYMRMPAS 8.2 IC50 2
FEZYZPVXOKHVHG 8.2 Ki 3
MUMWTBPFGOZRHX 8.2 Ki 3
NBMJTOOHXJGJNZ 8.2 Ki 2
NTNRVRBIIZBTBR 8.2 IC50 8
NVRLHRULRRIJBY 8.2 Ki 3
QPLOFYKBIFMXBX 8.2 IC50 2
VVPIFAABYQQPKY 8.2 IC50 2
DNNZYGQJIKJSHH 8.1 IC50 3
LARGKTWCHAEXEF 8.1 IC50 2
OUOIBTWZEMQDJD 8.1 IC50 2
FDLUVBKZNIPEQR 8.1 Ki 6
LZHGUODYTWJFHC 8.1 IC50 2
NJNGYXSQUSGZGO 8.1 IC50 2
OBSGJFCIYCQJEU 8.1 Ki 3
RMNQUVGQJWBXRY 8.1 IC50 2
XWIQXLQKQCPYLC 8.1 Ki 2
ZTJVQQCXGUIYTL 8.1 Ki 4
DGSNYQOOWLOGKI 8.1 Ki 3
MKSVLCRJUVAEQS 8.1 IC50 2
QENGYZQWMBJJRV 8.1 Ki 3
YNXCWDXRPDZZLO 8.1 IC50 2
DAZKRYLEGWSBDU 8.1 Ki 2
DWMRZXZBTGUNST 8.1 Ki 2
FXLFNEVHWHPROF 8.1 Ki 2
UZTAEKUHQOCYGB 8.1 Ki 3
VWSZBXMMCLLXFO 8.1 IC50 2
YGFGZLKRXRBORE 8.1 Ki 3
UAHXABWWDRJQRK 8.1 IC50 2
FRFVLJZLTVYZKB 8.1 IC50 2
2D structure