Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TZKJUKFMINMKSP
|
8.3 | IC50 | 2 | — | |
FQMWRNFRVKBREN
|
8.3 | IC50 | 2 | — | |
PDUMJXCNOKHQKH
|
8.3 | Ki | 9 | — | |
RMNQUVGQJWBXRY
|
8.3 | IC50 | 2 | — | |
SNUMNATTXKTJQD
|
8.3 | IC50 | 2 | — | |
IACDYBNAKZUROA
|
8.3 | IC50 | 2 | — | |
MSUOXKMCLUJSJC
|
8.3 | IC50 | 2 | — | |
QBWXHIMIUSZAOP
|
8.3 | IC50 | 2 | — | |
QELFRIHVHVRUFC
|
8.3 | IC50 | 2 | — | |
XSYGTWRAAARAFS
|
8.3 | IC50 | 2 | — | |
KZXNHUNTABHMLN
|
8.3 | Ki | 3 | — | |
LLNQIULEMBGSKZ
|
8.3 | IC50 | 2 | — | |
SATGRGDFTKEDOC
|
8.3 | IC50 | 2 | — | |
WVQIDDPAQZTNTF
|
8.3 | IC50 | 2 | — | |
YRUPTYVLRUXKLT
|
8.3 | IC50 | 2 | — | |
AITUBRIGGLTKMQ
|
8.3 | IC50 | 2 | — | |
BHHIIHJGDBVRNZ
|
8.3 | Ki | 3 | — | |
IOLSRAXZCKDSPO
|
8.3 | Ki | 6 | — | |
NEHLLAYKPWEYRL
|
8.3 | Ki | 3 | — | |
OLELYTACRIKUHK
|
8.3 | IC50 | 2 | — | |
QFJOOWSJASQPAX
|
8.3 | IC50 | 7 | — | |
QMPSRRLYDPGUKS
|
8.3 | Ki | 3 | — | |
VLNBINQYXHFUGN
|
8.3 | IC50 | 2 | — | |
VZCFMFWKMXXTFA
|
8.3 | Ki | 3 | — | |
VZEPGFGHCQNEFC
|
8.3 | IC50 | 2 | — | |
XATHBXYKVIAZOR
|
8.3 | Ki | 3 | — | |
XPDGYJOFZSUFCY
|
8.3 | IC50 | 2 | — | |
FUNCNRULOWTKJU
|
8.3 | IC50 | 2 | — | |
PGRXFTCYMWPHKW
|
8.3 | Ki | 2 | — | |
RUUQARAMINJWGP
|
8.3 | Ki | 2 | — | |
YXQQDNTZJAXMNL
|
8.3 | IC50 | 2 | — | |
FPAKZDLGEHHCTC
|
8.3 | IC50 | 2 | — | |
ZXSDTWYIYKNDSR
|
8.3 | IC50 | 2 | — | |
NPKCSHLGQLVUNO
|
8.2 | Ki | 3 | — | |
NYQZRXFSTDWBHC
|
8.2 | Ki | 2 | — | |
YGFSDBVKNXCHFA
|
8.2 | IC50 | 2 | — | |
AKWQVFJCPSUJBC
|
8.2 | IC50 | 2 | — | |
SBXOMGIKOINZME
|
8.2 | IC50 | 2 | — | |
UDQDURKQOJZYOA
|
8.2 | IC50 | 2 | — | |
UUUYIBUJURRXLR
|
8.2 | Ki | 3 | — | |
XYWIPYBIIRTJMM
|
8.2 | IC50 | 2 | — | |
MZJDBIVMBJLQSX
|
8.2 | IC50 | 2 | — | |
OEMBYSUFEIJUEQ
|
8.2 | IC50 | 2 | — | |
CIBAUUPUKBYRIO
|
8.2 | IC50 | 2 | — | |
DBBPDYZRKMIZOJ
|
8.2 | IC50 | 2 | — | |
GTOBEZUWBRGMLK
|
8.2 | IC50 | 2 | — | |
GZODXKWDFODGHQ
|
8.2 | Ki | 3 | — | |
HVNXYZZCSQONQC
|
8.2 | Ki | 2 | — | |
IEAPTAHBSJIEKO
|
8.2 | IC50 | 3 | — | |
JVCAULOQATWKKF
|
8.2 | IC50 | 2 | — |