Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORHCDONRNQJSDU
|
8.5 | IC50 | 2 | — | |
XMGACJAVDNSYFS
|
8.5 | IC50 | 2 | — | |
WBUMTRVFJVGNEX
|
8.5 | IC50 | 2 | — | |
HQFBMTXLTXVRAL
|
8.5 | IC50 | 2 | — | |
OXHLIVRHOPCUSV
|
8.5 | Ki | 5 | — | |
QNXVSHDBEGAVAR
|
8.5 | Ki | 3 | — | |
UAHXABWWDRJQRK
|
8.5 | IC50 | 2 | — | |
VFCPFXPPJSVUEB
|
8.5 | IC50 | 2 | — | |
NKCIMLZZOJBOGZ
|
8.5 | IC50 | 2 | — | |
QYWRPJPBRRCNJD
|
8.5 | Ki | 3 | — | |
AZBFGOGAJPTZRR
|
8.5 | IC50 | 2 | — | |
CGRKOXZKWKCFAG
|
8.5 | IC50 | 2 | — | |
LIFWZDTWISKRBJ
|
8.5 | Ki | 3 | — | |
CJLPNFNSEYZOKO
|
8.5 | IC50 | 2 | — | |
METWKYXLYOAEDA
|
8.5 | IC50 | 2 | — | |
QGNJMTPKSKWTBQ
|
8.5 | IC50 | 2 | — | |
UENKHDMGQRVXOA
|
8.5 | IC50 | 2 | — | |
VGEIARNAACQQRK
|
8.5 | IC50 | 2 | — | |
YXQQDNTZJAXMNL
|
8.5 | IC50 | 2 | — | |
ZYCBZVOBLYDGQZ
|
8.4 | IC50 | 2 | — | |
FTLCKEYXULODRH
|
8.4 | IC50 | 2 | — | |
JKKGBKZFKPXHDS
|
8.4 | Ki | 3 | — | |
KVALJOXTMDVFNN
|
8.4 | IC50 | 2 | — | |
UOFFBMYRFFCNLY
|
8.4 | IC50 | 2 | — | |
UOFFBMYRFFCNLY
|
8.4 | IC50 | 2 | — | |
CZWHJSKWMSOPRC
|
8.4 | IC50 | 2 | — | |
JREFSUNTZCXDKL
|
8.4 | IC50 | 2 | — | |
AJXCDVGDMKCSJV
|
8.4 | IC50 | 2 | — | |
DAVIKZRXBAXBIC
|
8.4 | IC50 | 2 | — | |
FAUPYRQOQINXOL
|
8.4 | IC50 | 2 | — | |
QWJAHBCIMJSNPO
|
8.4 | IC50 | 2 | — | |
YGSSAEZAISFQSW
|
8.4 | IC50 | 2 | — | |
DZZRWRHLIZMWFJ
|
8.4 | Ki | 3 | — | |
FVOIRKKFLDCVKH
|
8.4 | IC50 | 2 | — | |
KMNWQMKSCBCXNX
|
8.4 | Ki | 3 | — | |
BVZHCUOVJATBQP
|
8.4 | Ki | 5 | — | |
DUTABFFYBPSPBP
|
8.4 | IC50 | 6 | — | |
FSWZRDMSLCEJGG
|
8.4 | Ki | 3 | — | |
KJPOONPDKYPIKE
|
8.4 | Ki | 3 | — | |
MOLMATGEEFSJHI
|
8.4 | Ki | 3 | — | |
OWBNSFCRELNSPK
|
8.4 | Ki | 3 | — | |
WNBXSHDGFJUTNR
|
8.4 | Ki | 2 | — | |
WYOJURVOHOBMRY
|
8.4 | Ki | 2 | — | |
YDTFCSKLISVNDE
|
8.4 | Ki | 3 | — | |
ZDMYKWNIEWNTLR
|
8.4 | IC50 | 5 | — | |
KNUYTWQBCBAZFL
|
8.4 | IC50 | 2 | — | |
XMCZMUIHYCVFKG
|
8.4 | Ki | 2 | — | |
ZAKSQHPNZWUBFJ
|
8.4 | IC50 | 2 | — | |
AWJUPCORVZXGJV
|
8.4 | IC50 | 2 | — | |
JFTPUCJHGXFNAL
|
8.4 | IC50 | 2 | — |