Target Details
UniProt ACP03952
Gene SymbolKLKB1
Protein NamePlasma kallikrein
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00024 (PAN_1) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,277
  • Clinical molecules 0
  • Avg pChEMBL 7.55
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,277)
InChIKey pChEMBL Type Targets Clinical
ORHCDONRNQJSDU 8.5 IC50 2
XMGACJAVDNSYFS 8.5 IC50 2
WBUMTRVFJVGNEX 8.5 IC50 2
HQFBMTXLTXVRAL 8.5 IC50 2
OXHLIVRHOPCUSV 8.5 Ki 5
QNXVSHDBEGAVAR 8.5 Ki 3
UAHXABWWDRJQRK 8.5 IC50 2
VFCPFXPPJSVUEB 8.5 IC50 2
NKCIMLZZOJBOGZ 8.5 IC50 2
QYWRPJPBRRCNJD 8.5 Ki 3
AZBFGOGAJPTZRR 8.5 IC50 2
CGRKOXZKWKCFAG 8.5 IC50 2
LIFWZDTWISKRBJ 8.5 Ki 3
CJLPNFNSEYZOKO 8.5 IC50 2
METWKYXLYOAEDA 8.5 IC50 2
QGNJMTPKSKWTBQ 8.5 IC50 2
UENKHDMGQRVXOA 8.5 IC50 2
VGEIARNAACQQRK 8.5 IC50 2
YXQQDNTZJAXMNL 8.5 IC50 2
ZYCBZVOBLYDGQZ 8.4 IC50 2
FTLCKEYXULODRH 8.4 IC50 2
JKKGBKZFKPXHDS 8.4 Ki 3
KVALJOXTMDVFNN 8.4 IC50 2
UOFFBMYRFFCNLY 8.4 IC50 2
UOFFBMYRFFCNLY 8.4 IC50 2
CZWHJSKWMSOPRC 8.4 IC50 2
JREFSUNTZCXDKL 8.4 IC50 2
AJXCDVGDMKCSJV 8.4 IC50 2
DAVIKZRXBAXBIC 8.4 IC50 2
FAUPYRQOQINXOL 8.4 IC50 2
QWJAHBCIMJSNPO 8.4 IC50 2
YGSSAEZAISFQSW 8.4 IC50 2
DZZRWRHLIZMWFJ 8.4 Ki 3
FVOIRKKFLDCVKH 8.4 IC50 2
KMNWQMKSCBCXNX 8.4 Ki 3
BVZHCUOVJATBQP 8.4 Ki 5
DUTABFFYBPSPBP 8.4 IC50 6
FSWZRDMSLCEJGG 8.4 Ki 3
KJPOONPDKYPIKE 8.4 Ki 3
MOLMATGEEFSJHI 8.4 Ki 3
OWBNSFCRELNSPK 8.4 Ki 3
WNBXSHDGFJUTNR 8.4 Ki 2
WYOJURVOHOBMRY 8.4 Ki 2
YDTFCSKLISVNDE 8.4 Ki 3
ZDMYKWNIEWNTLR 8.4 IC50 5
KNUYTWQBCBAZFL 8.4 IC50 2
XMCZMUIHYCVFKG 8.4 Ki 2
ZAKSQHPNZWUBFJ 8.4 IC50 2
AWJUPCORVZXGJV 8.4 IC50 2
JFTPUCJHGXFNAL 8.4 IC50 2
2D structure