Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KPFQKUFJYSBYBL
|
8.5 | IC50 | 3 | — | |
KPLOPAOSJILVIG
|
8.5 | IC50 | 4 | — | |
LAEZPLWSRMVDKT
|
8.5 | IC50 | 5 | — | |
MBBRYSHFZAKDNK
|
8.5 | Ki | 3 | — | |
NDQYBUYVXIWGNJ
|
8.5 | IC50 | 3 | — | |
NFRBICAIEMTSJZ
|
8.5 | Ki | 2 | — | |
NTFAJFSJGVPGAC
|
8.5 | IC50 | 3 | — | |
OGEBHANRXXUPQA
|
8.5 | IC50 | 3 | — | |
OITRKHUOZGPBJI
|
8.5 | Ki | 4 | — | |
OJOAPDZWILJFFF
|
8.5 | IC50 | 2 | — | |
ONIHHUWDVFUCAR
|
8.5 | Ki | 3 | — | |
OQHYZXMZPSUAEY
|
8.5 | IC50 | 7 | — | |
OTZKOBJGNWYHCY
|
8.5 | IC50 | 3 | — | |
PHLLDHUJAMWXHD
|
8.5 | IC50 | 3 | — | |
PIUDHEFNICCZME
|
8.5 | IC50 | 2 | — | |
PIUDHEFNICCZME
|
8.5 | IC50 | 2 | — | |
QCLWJMUFTKLIAE
|
8.5 | IC50 | 2 | — | |
QFJLWQWOKYLTEQ
|
8.5 | Ki | 3 | — | |
QKUJFWQNWXUDGB
|
8.5 | IC50 | 2 | — | |
QSWJYWCLHVAJEZ
|
8.5 | IC50 | 2 | — | |
RGZWSMZUUVHSMD
|
8.5 | IC50 | 3 | — | |
RJGXWYMMSWXDBY
|
8.5 | IC50 | 4 | — | |
RJQLFWVERDFMFU
|
8.5 | IC50 | 4 | — | |
RMNYKKOMVGKWMF
|
8.5 | IC50 | 3 | — | |
RRDABEWIPOYJNA
|
8.5 | IC50 | 2 | — | |
RWQRQTTUCTXRQC
|
8.5 | IC50 | 4 | — | |
SAQOYLCNEVUQKH
|
8.5 | IC50 | 3 | — | |
SBFVHGJSVOMQJH
|
8.5 | IC50 | 4 | — | |
SJKSASQLXWHGFH
|
8.5 | IC50 | 4 | — | |
SUNUOUSWUILJOO
|
8.5 | Ki | 3 | — | |
SVWVNWWLYZGNGT
|
8.5 | IC50 | 2 | — | |
SWVWAZLEARISBG
|
8.5 | IC50 | 2 | — | |
SXIFTOXSOJHIGC
|
8.5 | IC50 | 3 | — | |
SXVRJEWRROULBO
|
8.5 | IC50 | 4 | — | |
UPPRVHQOSXWZLP
|
8.5 | IC50 | 3 | — | |
VARXLQCHRPURJT
|
8.5 | IC50 | 3 | — | |
VFEVHMYHGBXCLM
|
8.5 | IC50 | 3 | — | |
WJAIHAMGHSKLNB
|
8.5 | IC50 | 2 | — | |
WMVZLWYOHAUGMC
|
8.5 | IC50 | 3 | — | |
WQVBAYOMZJYFJK
|
8.5 | IC50 | 8 | — | |
WUPABZDGAQQKAU
|
8.5 | Ki | 3 | — | |
WZFGKOMTANPZBQ
|
8.5 | IC50 | 2 | — | |
XGBLRGJOWPDUDW
|
8.5 | IC50 | 3 | — | |
XQRKYMOJJOXHBZ
|
8.5 | IC50 | 2 | — | |
YBAIRJKLWQYRGC
|
8.5 | IC50 | 2 | — | |
YCUHYXGBQOXOJG
|
8.5 | IC50 | 6 | — | |
YHMGDTWUZGOVRL
|
8.5 | IC50 | 2 | — | |
YSHBWHHQCNCYQM
|
8.5 | IC50 | 2 | — | |
ZKYUOZOXYNXLAA
|
8.5 | IC50 | 4 | — | |
DUPDRBCVCXMPPE
|
8.5 | Ki | 3 | — |