Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LQEJGKWBOTZIBV
|
8.6 | IC50 | 2 | — | |
PQLJHTCQQFICKU
|
8.6 | IC50 | 2 | — | |
QMJWWNVVTLEZIW
|
8.6 | Ki | 3 | — | |
SADGBXCCQGIXDH
|
8.6 | IC50 | 2 | — | |
UDQDURKQOJZYOA
|
8.6 | IC50 | 2 | — | |
ARIOOOOXKGGXCY
|
8.6 | IC50 | 2 | — | |
SOLNGYFEBLRSAN
|
8.6 | IC50 | 2 | — | |
ZIAUCGPBMPJNBL
|
8.6 | IC50 | 2 | — | |
GEDGCUQVJCWBFY
|
8.6 | IC50 | 2 | — | |
SATGRGDFTKEDOC
|
8.6 | IC50 | 2 | — | |
VNKFZBCCJJVXJG
|
8.6 | Ki | 5 | — | |
NINJGBVHUFUANQ
|
8.6 | IC50 | 2 | — | |
AZYMEDAZJNOBLR
|
8.5 | IC50 | 2 | — | |
BKOMRHGWSXFZSH
|
8.5 | IC50 | 3 | — | |
KXLAWRVDSZAFKG
|
8.5 | IC50 | 2 | — | |
NAHGIMDHYQSLEN
|
8.5 | Ki | 2 | — | |
XMXXHDVGILDRBZ
|
8.5 | IC50 | 2 | — | |
OCWLBXWNNDGCER
|
8.5 | Ki | 3 | — | |
ABVVTLDDAJPMKZ
|
8.5 | IC50 | 3 | — | |
AJQGZKKQAAWAPQ
|
8.5 | IC50 | 6 | — | |
AKZWUAZVOXSXOH
|
8.5 | Ki | 3 | — | |
AQESQZZCMQJOJU
|
8.5 | Ki | 2 | — | |
ASPQAQDFTSKEAM
|
8.5 | IC50 | 2 | — | |
BKGCNONNVNNPCJ
|
8.5 | IC50 | 2 | — | |
BYCWLOQDZYMODR
|
8.5 | Ki | 3 | — | |
COGDLYORVLPAJK
|
8.5 | IC50 | 3 | — | |
CQDVUJSXYFSSHR
|
8.5 | IC50 | 4 | — | |
CSOIEWKCRIAOFP
|
8.5 | IC50 | 2 | — | |
CUJAMZMFVUMLMN
|
8.5 | IC50 | 3 | — | |
DHWRFOFVRNXWFE
|
8.5 | IC50 | 2 | — | |
DVKBAFOJFMJCAO
|
8.5 | IC50 | 2 | — | |
DVMDKOVGIYJULU
|
8.5 | IC50 | 4 | — | |
DXCOONBXASCQJO
|
8.5 | IC50 | 4 | — | |
FCXNRNCBQJLWDJ
|
8.5 | IC50 | 3 | — | |
FTZQENZGWYGYSA
|
8.5 | IC50 | 2 | — | |
FUQWXNUBICSJBF
|
8.5 | IC50 | 4 | — | |
FXBYCOIBSNRTHQ
|
8.5 | Ki | 2 | — | |
GANUYKJXFODNNH
|
8.5 | IC50 | 2 | — | |
GBMNOBITEYOELC
|
8.5 | IC50 | 2 | — | |
GLWZFGZVOWCXPQ
|
8.5 | IC50 | 2 | — | |
GZIWAJRNQSUBEG
|
8.5 | Ki | 3 | — | |
GZWDTTNGXUYGCU
|
8.5 | IC50 | 3 | — | |
IEVMGHWIRRVDRB
|
8.5 | Ki | 3 | — | |
IIHKCWBLAFVPAV
|
8.5 | IC50 | 2 | — | |
JBHALIPUGWBOFZ
|
8.5 | IC50 | 2 | — | |
JIRZTKNHLRBCKF
|
8.5 | IC50 | 3 | — | |
JIRZTKNHLRBCKF
|
8.5 | IC50 | 3 | — | |
JSZAYFVPBHXVCY
|
8.5 | Ki | 3 | — | |
KITXJRBAWLMDQM
|
8.5 | IC50 | 3 | — | |
KKQBOZNOYSOFLO
|
8.5 | Ki | 3 | — |