Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RRYHCECMCWJEIU
|
8.8 | Ki | 3 | — | |
ZXSDTWYIYKNDSR
|
8.8 | IC50 | 2 | — | |
GTZXEPXZPDKLLW
|
8.8 | IC50 | 2 | — | |
FVOIRKKFLDCVKH
|
8.8 | IC50 | 2 | — | |
IQNORUMXNDXEIL
|
8.8 | IC50 | 2 | — | |
IQNORUMXNDXEIL
|
8.8 | IC50 | 2 | — | |
OEMBYSUFEIJUEQ
|
8.8 | IC50 | 2 | — | |
ZJYAXUISSVXYQC
|
8.8 | IC50 | 2 | — | |
HOSBKCRSFCXIDE
|
8.8 | IC50 | 2 | — | |
FCSAYDZPMDLFSN
|
8.7 | IC50 | 2 | — | |
NZYSNSQHJHYDEI
|
8.7 | IC50 | 2 | — | |
OPAHIKCMESQWDF
|
8.7 | IC50 | 2 | — | |
QEBKYPAJRRRDKH
|
8.7 | IC50 | 2 | — | |
WSCJCNZPEVIQIK
|
8.7 | IC50 | 2 | — | |
ZOIAMJPHWFPPNK
|
8.7 | IC50 | 2 | — | |
UHRURUXVXNFGPR
|
8.7 | IC50 | 2 | — | |
AWLPKPUSDZNVQR
|
8.7 | IC50 | 2 | — | |
GAVRMVQHHVMXFD
|
8.7 | Ki | 11 | — | |
KNJDMNATKQSVKK
|
8.7 | IC50 | 2 | — | |
XCJQHVXBYDODIH
|
8.7 | IC50 | 3 | — | |
BOCSUPFQLFIHFX
|
8.7 | IC50 | 4 | — | |
FANJUXPUAIHWDE
|
8.7 | IC50 | 5 | — | |
FDORZCAYZLDCPZ
|
8.7 | Ki | 2 | — | |
GWZGMZVWURNLOZ
|
8.7 | Ki | 4 | — | |
HKBDZTCNUODKEC
|
8.7 | IC50 | 3 | — | |
LEOZSBNDFVBQQT
|
8.7 | IC50 | 5 | — | |
LRJDBUKQKSAXJD
|
8.7 | Ki | 3 | — | |
NKFYMWBVMOGCMS
|
8.7 | IC50 | 2 | — | |
OGCGKERBEQPTBU
|
8.7 | Ki | 3 | — | |
PDUMJXCNOKHQKH
|
8.7 | Ki | 4 | — | |
PKASBNFVFWUNOA
|
8.7 | IC50 | 4 | — | |
QCJKXYYLKAMQSD
|
8.7 | Ki | 5 | — | |
SRKDCGUSWAONMJ
|
8.7 | IC50 | 3 | — | |
URTZZBQNKCNCOJ
|
8.7 | Ki | 3 | — | |
UWCHLKPJXDNUJJ
|
8.7 | Ki | 3 | — | |
XRRSNWWFDKBFCV
|
8.7 | Ki | 3 | — | |
YCPIFMNZNHRZMY
|
8.7 | Ki | 3 | — | |
ZTXALZIIFRKUGE
|
8.7 | Ki | 3 | — | |
CYVJFYJEJKTVCI
|
8.7 | IC50 | 2 | — | |
HNHBZVLOAXVGOW
|
8.7 | IC50 | 2 | — | |
LHPWAHFZZCZBHC
|
8.7 | IC50 | 2 | — | |
QBWXHIMIUSZAOP
|
8.7 | IC50 | 2 | — | |
VQBUYPWHWZACJN
|
8.7 | IC50 | 2 | — | |
YYLJKEYIZVRFEV
|
8.7 | IC50 | 2 | — | |
SADGBXCCQGIXDH
|
8.7 | IC50 | 2 | — | |
HWKYPMGUMIKDKT
|
8.6 | Ki | 3 | — | |
YTULCQGNUIGFGU
|
8.6 | Ki | 2 | — | |
LJVRVBNTOCCTEO
|
8.6 | Ki | 2 | — | |
BKSCOHJNKDJECO
|
8.6 | Ki | 3 | — | |
GJQARFAKHMCMDU
|
8.6 | Ki | 2 | — |