Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CXCGNTAXXPYSAK
|
9.0 | Ki | 2 | — | |
GOERAAJVARXHDP
|
9.0 | IC50 | 4 | — | |
GTVFMNZALGQANW
|
9.0 | IC50 | 2 | — | |
HECONMODEBIAKY
|
9.0 | IC50 | 9 | — | |
HLWOCEXYCJLWGO
|
9.0 | Ki | 3 | — | |
HMMQIOFQLZWHKO
|
9.0 | IC50 | 2 | — | |
MAMDUCKALBRXSZ
|
9.0 | IC50 | 2 | — | |
MBFJFSDXDXLAQN
|
9.0 | IC50 | 2 | — | |
NDQYBUYVXIWGNJ
|
9.0 | IC50 | 2 | — | |
NDQYBUYVXIWGNJ
|
9.0 | IC50 | 2 | — | |
PKASBNFVFWUNOA
|
9.0 | IC50 | 2 | — | |
QUNVBYGAKUPYEF
|
9.0 | Ki | 3 | — | |
RDZCPPLNBZHPMQ
|
9.0 | Ki | 3 | — | |
SEYYELZSACSHCW
|
9.0 | Ki | 3 | — | |
VSUYWTSSABVZTL
|
9.0 | Ki | 3 | — | |
WIOGTPFOPDWSIT
|
9.0 | Ki | 3 | — | |
WNNVCOPVUBHDRW
|
9.0 | Ki | 3 | — | |
WSDKNZUBTLXSPM
|
9.0 | Ki | 3 | — | |
XXPYQZDZFMYLHR
|
9.0 | Ki | 3 | — | |
ZGZPKQSHBQJIGW
|
9.0 | IC50 | 2 | — | |
DXPRVTLHVRYGPT
|
9.0 | Ki | 2 | — | |
DROSFHKHAAIBHD
|
9.0 | IC50 | 2 | — | |
IMCXJEIDVWMIBG
|
9.0 | Ki | 3 | — | |
MUXOTMXNFWFKTR
|
9.0 | IC50 | 2 | — | |
UUIHUWPHJJSKFX
|
9.0 | IC50 | 2 | — | |
QZLHOCXIFYJRGS
|
8.9 | IC50 | 2 | — | |
GIVXPUNNLANRCG
|
8.9 | IC50 | 2 | — | |
XHOSJSGSUAYWPH
|
8.9 | IC50 | 2 | — | |
AEJZMQKSVVZBAW
|
8.9 | IC50 | 2 | — | |
KPLREYDSVWITHB
|
8.9 | IC50 | 2 | — | |
CYUSFSQPVJASKS
|
8.9 | IC50 | 2 | — | |
CZWHJSKWMSOPRC
|
8.9 | IC50 | 2 | — | |
DTIUMOLBWQXRPH
|
8.9 | Ki | 3 | — | |
RVENPILMUUNNIX
|
8.9 | IC50 | 2 | — | |
MNHRZKFGCZXRJO
|
8.9 | IC50 | 2 | — | |
WCNRFBOCXRIWNE
|
8.9 | IC50 | 2 | — | |
AEBJMLIAWHLLQF
|
8.9 | IC50 | 2 | — | |
AZYMEDAZJNOBLR
|
8.8 | IC50 | 2 | — | |
IAWTUPZVMCVDDL
|
8.8 | IC50 | 2 | — | |
IICMIKXBIINPOO
|
8.8 | IC50 | 2 | — | |
ORRIMSVBDDRCMC
|
8.8 | IC50 | 2 | — | |
QMYPKRMOPLSDIX
|
8.8 | IC50 | 2 | — | |
OCRCHYZWRKVQCQ
|
8.8 | IC50 | 2 | — | |
RZUBKNRJNSMNNO
|
8.8 | IC50 | 2 | — | |
BJLPPNMAKGCMOT
|
8.8 | IC50 | 2 | — | |
BJSIWIFJSRFHPS
|
8.8 | Ki | 6 | — | |
DVTLDIPPLKDTBX
|
8.8 | IC50 | 2 | — | |
MCDKKKIUEGNSPK
|
8.8 | Ki | 5 | — | |
QWJAHBCIMJSNPO
|
8.8 | IC50 | 2 | — | |
QWMGKGHSOYXEJP
|
8.8 | Ki | 3 | — |