Target Details
| UniProt AC | P03952 |
|---|---|
| Gene Symbol | KLKB1 |
| Protein Name | Plasma kallikrein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00024 (PAN_1) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,277
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BHQDUYVBGREBCB
|
10.7 | Ki | 8 | — | |
HEKNEXYMJKVOGQ
|
10.7 | Ki | 4 | — | |
HJCCPKALMCCVEK
|
10.1 | Ki | 5 | — | |
RCVRHAVSXLQPDX
|
10.1 | Ki | 5 | — | |
QTEIOTHWOLEZKV
|
10.0 | IC50 | 2 | — | |
XGUFEENWPFGFKD
|
10.0 | Ki | 2 | — | |
DCLSJFXDVAAQJQ
|
9.7 | IC50 | 2 | — | |
LQUYFWRKFWJAJB
|
9.7 | IC50 | 2 | — | |
ZAICGYJCCFAMHG
|
9.7 | IC50 | 2 | — | |
CUGMKURPXUMGSV
|
9.6 | Ki | 4 | — | |
AESNDDHBSPWNAX
|
9.5 | IC50 | 2 | — | |
DIFGLRSYVDIDJS
|
9.5 | Ki | 3 | — | |
VGFJEINHJGJRSC
|
9.5 | IC50 | 2 | — | |
HDFVEEOQSFUVTL
|
9.5 | IC50 | 2 | — | |
DKUIMPNNWCHYFQ
|
9.4 | IC50 | 2 | — | |
SHZUCTHKVWMOJI
|
9.4 | IC50 | 2 | — | |
ZOIAMJPHWFPPNK
|
9.4 | IC50 | 2 | — | |
DGIRMJAUTLUPMU
|
9.3 | IC50 | 2 | — | |
FUSZQUYKUCNCED
|
9.3 | IC50 | 2 | — | |
PCSCBPUPCOBODL
|
9.3 | IC50 | 2 | — | |
OTRDMMCGPKTUCO
|
9.3 | IC50 | 2 | — | |
QWRMLYGJHYOEIN
|
9.3 | IC50 | 2 | — | |
GWIGRUFPKOTEAQ
|
9.2 | Ki | 3 | — | |
UCJSXODQQLYFFF
|
9.2 | IC50 | 2 | — | |
BSNRZZUTVDCZAA
|
9.2 | IC50 | 2 | — | |
DKUIMPNNWCHYFQ
|
9.2 | IC50 | 2 | — | |
OUGUMFKJMHXPKT
|
9.2 | Ki | 2 | — | |
KVJUZBSCFYFGMJ
|
9.2 | IC50 | 2 | — | |
CEOSELUUHJNGPA
|
9.2 | IC50 | 2 | — | |
MRERGFSFJIIPPV
|
9.2 | IC50 | 3 | — | |
NHHYXMBQJKVFNB
|
9.2 | IC50 | 2 | — | |
BVIDABUHKFIJPH
|
9.1 | IC50 | 2 | — | |
DVMWQVLBMQQBHU
|
9.1 | IC50 | 2 | — | |
XCOPLNVIDMHZTN
|
9.1 | IC50 | 2 | — | |
GSFPQMPKJFXLTO
|
9.1 | IC50 | 2 | — | |
BHKJUCWCWRSZFB
|
9.1 | IC50 | 2 | — | |
DROSFHKHAAIBHD
|
9.1 | IC50 | 2 | — | |
SAULAGCQOSOMSG
|
9.1 | IC50 | 2 | — | |
HWYRMCCHOBIHJO
|
9.1 | IC50 | 2 | — | |
MNXBWEWRFDRXBD
|
9.1 | IC50 | 2 | — | |
SOARPTXSWUKGOA
|
9.1 | IC50 | 2 | — | |
BAVINDCBMIUDHY
|
9.1 | IC50 | 2 | — | |
LWFLIRIWEPBXFX
|
9.1 | Ki | 4 | — | |
OYUAZKUQDXYHFK
|
9.1 | IC50 | 2 | — | |
OZSFFGZNHVNMND
|
9.1 | IC50 | 2 | — | |
BSNRZZUTVDCZAA
|
9.0 | IC50 | 2 | — | |
AIRGERSZASMAFK
|
9.0 | IC50 | 2 | — | |
BAQBTVHTGIAQPV
|
9.0 | Ki | 3 | — | |
BPYVSZXRXGLXFP
|
9.0 | Ki | 3 | — | |
CSNSELBEUILYAV
|
9.0 | IC50 | 2 | — |