Target Details
UniProt ACP03369
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 70
  • Clinical molecules 0
  • Avg pChEMBL 8.59
Top Co-occurrence Targets
Active Molecules (70)
InChIKey pChEMBL Type Targets Clinical
UVTHAOVACKMIFO 7.5 Ki 2
HVXFNUXEOUIQKE 7.4 Ki 2
VEJOBLYVGLPABL 7.4 Ki 2
JBHCPNAOYVCBLC 7.4 Ki 2
BKVPEHBIRUOJPV 7.4 Ki 2
TUIJZRRAKRNJGG 7.4 Ki 2
ZMHLFTWXZHATIC 7.3 Ki 2
ZOGAJEOVCPKBPD 7.3 Ki 2
YTEURAFEAFHROU 7.3 Ki 2
XSHNENOGALPUOZ 7.1 Ki 2
HURZZMNNKMZLQC 7.0 Ki 2
XESKRTWBOYRKRZ 6.9 Ki 2
YZANKHXQXBZCRU 6.8 Ki 2
KDVFKVWSHSQULM 6.8 Ki 2
QBDOJPKXUDNOBE 6.8 Ki 2
KMGBJIFKTYDXGK 6.8 Ki 2
JBCCPGIVIKMXGT 6.7 Ki 2
LSEJXJJBPLLLBF 6.6 Ki 2
GQKWNYLKLDCKEF 6.5 Ki 2
RWBIVIUXFGDQLF 6.2 Ki 2
2D structure