Target Details
UniProt ACP03369
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 70
  • Clinical molecules 0
  • Avg pChEMBL 8.59
Top Co-occurrence Targets
Active Molecules (70)
InChIKey pChEMBL Type Targets Clinical
AIOQZNXKOQUMQK 10.8 Ki 2
IAINWMUGEQGIGE 10.8 Ki 2
LEJNWIFUYPPOMU 10.6 Ki 2
MUVGKQKGHIBGIU 10.5 Ki 2
WJOVSXDCDUIEBO 10.4 Ki 2
MRYXOBTXQMUTHQ 10.3 Ki 2
ZNYKWJFUQGHVRX 10.2 Ki 2
GOKNBQOQISRCDE 10.1 Ki 2
HWDFRZXEPANLKF 10.1 Ki 2
SLMZIXVIEWNEAM 10.1 Ki 3
NMHTYOAWRSWRPT 10.1 Ki 2
IGYIMSLYOKOAJR 10.0 Ki 3
JETOZULVKOQOTP 10.0 Ki 2
LLZSWFYHNNFIKA 9.9 Ki 2
LEJNWIFUYPPOMU 9.8 Ki 2
NEHGXHWAAYVUDY 9.8 Ki 2
YMARZQAQMVYCKC 9.8 Ki 6
OFOGUJVQCJTBKJ 9.7 Ki 2
QDJXSZXMSHHSJN 9.6 Ki 2
XETSHCIFFATMOX 9.6 Ki 2
ICLGGNKOSYUHKP 9.5 Ki 2
YAUPSJXHXSEEKT 9.5 Ki 2
KWVPZPFHKDDRKV 9.5 Ki 2
BUJKGFQFFGUYEM 9.4 Ki 2
GNJDFMNCMAQPGN 9.4 Ki 3
LAEBWIYUPGQNFS 9.4 Ki 2
ZMGRSVYTEJGXPC 9.3 Ki 2
PUSRVEPTERUAIU 9.2 Ki 2
ORFHUHJBECIJRM 9.1 Ki 2
RZCSYMCCZXFLPH 9.1 Ki 2
ZYGJIVAYVQHQAD 9.1 Ki 2
IKIBOJUXKVIMKQ 8.9 Ki 2
HVXFNUXEOUIQKE 8.9 Ki 3
CEVRDVWOXATASV 8.7 Ki 2
QQMKKKSPIWRIDH 8.7 Ki 2
LLSDCSYISTWPMW 8.6 Ki 2
GMZJLQXXVYHTRJ 8.6 Ki 2
XKWMIPNLKJFKLK 8.5 Ki 2
VHHGFQQTNGLIIJ 8.4 Ki 2
MVEFGMVKYUWSQO 8.1 Ki 2
ODZZSPNMADKGPQ 8.1 Ki 2
YYBURQAPOYNWBT 8.0 Ki 2
IGYIMSLYOKOAJR 8.0 Ki 2
KLUPNGHJEAUIGT 8.0 Ki 2
CZPLKLADANMGQQ 7.9 Ki 2
AGTAFMHGZWVOJS 7.9 Ki 2
XESKRTWBOYRKRZ 7.9 Ki 2
BFHBZKMCMTWBSI 7.7 Ki 2
JPSCLCKRSRMCFP 7.6 Ki 2
ZXHDUBIVQDVCIO 7.5 Ki 2
2D structure