Target Details
UniProt ACP03367
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 310
  • Clinical molecules 0
  • Avg pChEMBL 8.44
Top Co-occurrence Targets
Active Molecules (310)
InChIKey pChEMBL Type Targets Clinical
DESRIHHDJCUSEM 7.5 IC50 2
DRAQQTVGOMUDKD 7.5 Ki 2
FGLAXNOJEHONOE 7.5 Ki 2
GIMVBMLYXOBVGH 7.5 Ki 2
SSPOMXWWHDMCTH 7.5 Ki 2
DCGZDWXALWANQB 7.5 Ki 2
KUCPBPMVWXJNAI 7.5 Ki 2
ULBYZNDXPCBOLF 7.5 Ki 2
DESRIHHDJCUSEM 7.5 Ki 2
VYSKDMAUVBQCBE 7.4 Ki 2
FADBDGCGGLEUOC 7.4 Ki 2
PBWNGEMFPZKLHH 7.4 Ki 2
QNAMUDMCVZGMML 7.4 Ki 2
VBDZKMDDVRLKNW 7.4 Ki 2
YPUNDRMPWIYRAB 7.3 Ki 2
FTNYZEKSGWZDIC 7.3 Ki 2
JHFLECJGWVTYJX 7.3 Ki 2
XJRDHWPDPPVFPQ 7.3 Ki 2
GCGBTQJHRQVAMC 7.3 Ki 2
IJCXSYFOPRLLCZ 7.3 Ki 2
JWCCTWQEZATYNQ 7.3 Ki 2
ZDTGEVPZODCFNI 7.3 Ki 2
GXVFZTDCQPAGSZ 7.3 Ki 2
RBHLYDAZGYDJGN 7.3 Ki 2
SNBUCNNUZSAWLL 7.3 Ki 2
CWMBLJUBLZGJFU 7.2 Ki 2
HVCGCQVDUHANJA 7.2 Ki 2
VYANBIBLIUKGJH 7.2 Ki 2
PQJCVHDSBMYBNP 7.1 Ki 2
XVVVWGGOGOEGCN 7.1 Ki 2
DPLHSSKHQGEHNY 7.0 Ki 2
MPLBXHZCQCEEFQ 7.0 Ki 2
NOUUYGLUXBQXTQ 7.0 Ki 2
HIMYXPUMLAHVRJ 7.0 Ki 2
ITHMKJIOEXGHDG 7.0 Ki 2
LKCCOVZVNWPCLW 7.0 Ki 2
JTWDROYVKFPRKK 6.9 Ki 2
SFWDZUDCHHDDNN 6.9 Ki 2
LEQMLOFBCWZPIR 6.8 Ki 2
WHRABYWAWCKTGZ 6.8 Ki 2
MBGZGGPCRBOQQG 6.8 Ki 2
LLBMYBKLRLGOHL 6.7 Ki 2
SJDCULKXPKZGGR 6.7 Ki 2
SPFDDOLVNJYPAH 6.7 Ki 2
DOUAIUPZABTSSV 6.6 Ki 2
FSHUUSFSAWCFAT 6.6 Ki 2
YIZAIIPIDVPFIM 6.6 Ki 2
NPRGBQREGMCURE 6.6 Ki 2
OYNFRQIQIBKTHH 6.6 Ki 2
MMQQXXROQWAOCS 6.5 Ki 2
2D structure