Target Details
UniProt ACP03367
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 310
  • Clinical molecules 0
  • Avg pChEMBL 8.44
Top Co-occurrence Targets
Active Molecules (310)
InChIKey pChEMBL Type Targets Clinical
KVURTRGFRUMHJA 8.1 Ki 2
VSCUBCGPKBGSHX 8.1 Ki 2
KALBMBJPMINLKP 8.1 IC50 2
ZPHLTPTULPCICG 8.1 Ki 2
GMQJLAMTPFFOGB 8.0 Ki 2
BFUBIKTUZNMXLM 8.0 Ki 2
BJOKVXKYQNWVOS 8.0 Ki 2
BELVCNIPCAQSDE 8.0 Ki 2
SFXXPTJAVSRADD 8.0 Ki 2
OCCXDZCVCRGKNC 7.9 Ki 2
CRRZARJNNKORLN 7.9 Ki 2
ITMAELNBSPGPRZ 7.9 IC50 2
JIGPDMMPUDHDSE 7.9 Ki 2
UWJGSOBAFMJAGX 7.9 Ki 2
VNWDQLNHUXTPLV 7.9 Ki 2
WKMWOKUOGDUGMA 7.9 Ki 2
ZKWKOYXTTRVTSM 7.9 Ki 2
JZCAHOBXDOCSRW 7.9 IC50 2
SFIKZNVTYXSZBV 7.9 Ki 2
HPMPARPJICICTB 7.8 Ki 2
JNQDZKNQSKURFC 7.8 Ki 2
SXZREBMMGUVYHI 7.8 Ki 2
BKZLAIKLTFTJTM 7.8 Ki 2
CWMBLJUBLZGJFU 7.8 Ki 2
SUBZNMVLANXAJT 7.8 Ki 2
DKTCANLBUFELFO 7.8 Ki 2
POLWJEHKFDQFDZ 7.8 Ki 2
QUUQERMKKZCHEO 7.8 Ki 2
WPMSUJIOSJKBDT 7.8 Ki 2
ZQPMIVQPQJXWKF 7.8 Ki 2
YRGKHPCCNGDRSX 7.8 Ki 2
QENNGCUCJBLCNI 7.8 IC50 2
FXKDMLDFKKLUEV 7.8 Ki 2
FPCXMILVEIMFDV 7.7 Ki 2
VMAACENPBLBGNM 7.7 Ki 2
YWKIWUVMOWTVFX 7.7 Ki 2
WFVLXAJTZZDGIZ 7.7 Ki 2
URMXWTWEOOMAMJ 7.7 Ki 2
VRPYTXIQAZYPAK 7.7 Ki 2
SCPPGKSTBURNFW 7.7 Ki 2
XWDVRTHHZYSGAH 7.7 Ki 2
DVAMPQUOHXJGKH 7.7 Ki 2
GCANREIOWKPDFF 7.7 Ki 2
HWOINVSGNIWHKK 7.7 Ki 2
SFZSFNOTTPWXJH 7.6 Ki 2
WJNUCRCRECFEDH 7.6 Ki 2
ICAZGZKNGRQKPM 7.6 Ki 2
IZHOPUUPGTUJKC 7.6 Ki 2
BVXWMYQTUQMUTR 7.5 Ki 2
BLSNPKDSVTUIHC 7.5 Ki 2
2D structure