Target Details
UniProt ACP03367
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 310
  • Clinical molecules 0
  • Avg pChEMBL 8.44
Top Co-occurrence Targets
Active Molecules (310)
InChIKey pChEMBL Type Targets Clinical
GSKRTNPTDULYSS 8.4 Ki 2
WNFJASDZOJMGEK 8.4 Ki 2
WSIGESKMDUMSIL 8.4 Ki 2
BZXPRPQYBKHJGU 8.4 Ki 2
MGTJZTGXMAKEGV 8.4 Ki 2
NKZUVGNXYGUTGS 8.4 Ki 2
QZTNLTALZBMNPA 8.4 Ki 2
WRUVOSYKHXGAQN 8.4 Ki 2
ZMTSUDMDVPYUFD 8.4 Ki 2
HCFIPXMDHMTYDP 8.4 Ki 2
VMXVHXSZACZJHA 8.4 IC50 2
JETADCIDVOPMFX 8.3 Ki 2
TVXXCEMEGNEGDU 8.3 Ki 2
IWJSQELMWLOYSO 8.3 Ki 2
YKPHAYCUAMAQPA 8.3 Ki 2
WMJABJAWSXWQQI 8.3 Ki 2
MXZUOYJAKKUHJB 8.3 IC50 2
QMXOQNXRSPGBHU 8.3 Ki 2
UXBUYQULNOSYKV 8.3 Ki 2
AMVDOBISLYZBFC 8.3 Ki 2
DZUIVLUOOCSDIW 8.3 Ki 2
RCUVMESRLXGXNW 8.3 Ki 2
FTBLXBYPPSJOGB 8.3 Ki 2
RXFPKKNLUVRZTM 8.3 Ki 2
AYQCDKQNMGJQDP 8.2 Ki 2
VCEGGCOXLZWFIB 8.2 Ki 2
HROGQBIYFLWWNM 8.2 IC50 2
ZQTXOGGDJIFYFB 8.2 Ki 2
OZFMLABPBWLLNO 8.2 Ki 2
CULKWWDNMBXCFU 8.2 Ki 2
IMNORLPANFVGMK 8.2 Ki 2
YUZALEJJOXEEJU 8.2 IC50 3
VONDGXFKSSKVJE 8.2 Ki 2
DYBIOFGODCQGHH 8.2 Ki 2
BJSAKQUILVNYIK 8.2 Ki 2
CUWXKTMQEYYKBE 8.2 Ki 2
KVBJLSHFPVVAPU 8.2 Ki 2
WTDVMSFXXBREEA 8.2 Ki 2
ZQPMIVQPQJXWKF 8.2 Ki 2
FHWFGNNPLKNFPL 8.2 Ki 2
JUQPIABICJKAQY 8.2 IC50 2
LYOGIXRQACPKHV 8.2 Ki 2
NUVAAKOSCBUFEQ 8.2 Ki 2
POOYFSKIKCCODJ 8.2 IC50 2
OYQVQLRVPGEWPA 8.1 Ki 2
RVNBWRQFBXXQCM 8.1 Ki 2
XKOSXWLKHJUDDB 8.1 Ki 2
UWEBUXQKMPHDIG 8.1 Ki 2
WGNXTDDSGVECCL 8.1 Ki 2
BBVZGZMKVCDKNO 8.1 Ki 2
2D structure