Target Details
UniProt ACP03367
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 310
  • Clinical molecules 0
  • Avg pChEMBL 8.44
Top Co-occurrence Targets
Active Molecules (310)
InChIKey pChEMBL Type Targets Clinical
DCNBOHVQLTUPPO 8.8 Ki 2
FPWMFFCUHJOZBC 8.8 Ki 2
POZMOLJVHGBVQU 8.8 Ki 2
WIWOANAWRGKNSI 8.8 Ki 2
ZQCWCMLUKDMZGT 8.8 Ki 2
BTVVAWAWQSVPJK 8.8 Ki 2
XBQGRVOIPHJWJN 8.8 Ki 2
YDPDKRBSDWRYSP 8.8 Ki 2
PEUMBNRZJKVONR 8.8 Ki 2
SBGQHZJOYMMEFB 8.8 Ki 2
AYPUGIQXANZCKJ 8.7 Ki 2
RSIZVCJHRDDDBO 8.7 Ki 2
YMTOUOZOBVYCFQ 8.7 Ki 2
GOKWKRPSLDTITG 8.7 Ki 2
MSBYYCSXZCEAQC 8.7 Ki 2
NPRGBQREGMCURE 8.7 Ki 2
NPRGBQREGMCURE 8.7 IC50 2
RTLPHHSSFSSEFA 8.7 Ki 2
WPMLSGGBESQETR 8.7 Ki 2
FKDHOENKKMWEMD 8.7 Ki 2
LDJWKKOBSVJUAX 8.7 Ki 2
LUFAPAHVZKKIAU 8.7 Ki 2
YLZXTYZKINQZLV 8.7 Ki 2
MEMWZEJKDLLITJ 8.6 Ki 2
QIIKEDUNGZNOBB 8.6 Ki 2
WKDQVKFIFTZIHF 8.6 Ki 2
NPPRMIZPWNCEAK 8.6 Ki 2
PWTBXIFCEAJMHS 8.6 Ki 2
QYFVKQGRXSWYHA 8.6 Ki 2
RXURENWFZOYDPW 8.6 Ki 2
CBWQRQVEXJTNOT 8.6 Ki 2
RDJMIENHFLFNJX 8.6 Ki 2
WIJFQBUVCHIMHL 8.6 Ki 2
GQOPCFAFZYELPN 8.6 Ki 2
VRXKJOIIPJFAMB 8.6 Ki 2
JTEJMFKHUDDIBU 8.6 Ki 2
ZQTXOGGDJIFYFB 8.6 Ki 2
JOPONHSJMMHOPQ 8.5 Ki 2
UIJTVLDYMXSMIP 8.5 Ki 2
WKVNGPLMYBRORB 8.5 Ki 2
CZMAOEAHNYOMPV 8.5 IC50 2
DORNGHWKRMVHHU 8.5 Ki 2
RDXCKRVQYQGLCC 8.5 Ki 2
YIPXLIJTJWEEMN 8.5 Ki 2
KBIPGDRYFVMXGQ 8.5 Ki 2
GIKRNNJJZKPFLJ 8.5 Ki 2
QTIDFKQAHPGAQB 8.5 Ki 2
BPRDTHVBAHPJNR 8.4 Ki 2
IXHSGRWAMNNNRD 8.4 Ki 2
SPDFGCYXBCIFOC 8.4 Ki 2
2D structure