Target Details
UniProt ACP03367
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 310
  • Clinical molecules 0
  • Avg pChEMBL 8.44
Top Co-occurrence Targets
Active Molecules (310)
InChIKey pChEMBL Type Targets Clinical
FFUDEABEDNGPMU 9.5 Ki 2
VUYPJDFAKYXJEV 9.5 Ki 3
ZQTXOGGDJIFYFB 9.5 Ki 2
RHDRKQCNNGBNHC 9.5 Ki 2
SBKIEODZDWYACX 9.5 Ki 2
ROVMHUDIATYNMU 9.4 IC50 2
QHMBKCCJSCSGHG 9.4 Ki 3
HYNYUFZPPJMPOB 9.4 Ki 2
JRHBADZWYCWKNA 9.4 Ki 2
SCAKARIEFOIUDT 9.4 Ki 2
XZXHNGKWVNDCLC 9.3 Ki 2
KDHQYDMSHOTGOD 9.2 Ki 2
KBBBMHGFCVYISD 9.2 Ki 2
OOJVHJCVKLRBDZ 9.2 Ki 2
XISQZIYLHTUXPS 9.2 Ki 2
USPVZNGEOQQYLK 9.2 Ki 2
ZOQNQJASZAYUOG 9.2 Ki 2
JNIHRKHVDUSRFC 9.2 Ki 2
BOHAIUZINOMMEV 9.2 Ki 2
WNMJCUSDEYDSNU 9.1 Ki 2
NUZLDHGOBUOVBV 9.1 Ki 2
WALQPAXBTKJPQQ 9.1 Ki 2
NDYGPGKFUUCKOT 9.1 Ki 2
RMTJFBGMEPVVGM 9.1 Ki 2
PAUIHFDXSPYWNF 9.1 Ki 2
ZUJGJNYAFLLTGY 9.1 Ki 2
CGEAVTIBLIALNG 9.0 Ki 2
RVUHKVKFSGQQIN 9.0 Ki 2
WWTSWTPNILRSJX 9.0 Ki 2
QGDFPFVWJWQHNQ 9.0 Ki 2
BHIWBIFSAJDGCM 9.0 Ki 2
OSESYLJAMKLVDA 9.0 Ki 2
AJZAPEZJWWQJHC 8.9 Ki 2
BUEYISJFODTUIB 8.9 Ki 2
DVIKQNFIOVYHIX 8.9 Ki 2
HNWZJOSYFBXZFH 8.9 Ki 2
JWYLJKYZDLQQHI 8.9 Ki 3
QAGYKUNXZHXKMR 8.9 Ki 6
SMRBDAAALPUZDJ 8.9 Ki 2
IMVPEXQMZSPDQZ 8.9 Ki 2
ACIVSSKFPCODPQ 8.9 Ki 2
AFJXCHNRSQQDSV 8.8 Ki 2
CUSSQSVURRNYDL 8.8 Ki 2
DCQYMSCVLYZBBA 8.8 Ki 2
GNZIXCJETYMUQA 8.8 Ki 2
IKNWLZXHIFAHDB 8.8 Ki 2
IXMFJRZMSUIMQY 8.8 Ki 2
PMHSZNVAWHOHMK 8.8 Ki 2
UWMAWECJLCRQTB 8.8 Ki 2
XFXPDDPZRKCPBM 8.8 Ki 2
2D structure