Target Details
UniProt ACP03367
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 310
  • Clinical molecules 0
  • Avg pChEMBL 8.44
Top Co-occurrence Targets
Active Molecules (310)
InChIKey pChEMBL Type Targets Clinical
VYBDPVQMILRSMK 11.3 Ki 2
YOBNNQXGIZIFRK 11.0 Ki 2
BINXAIIXOUQUKC 10.8 Ki 3
XFNBBSJRWLSLFP 10.8 Ki 2
LTLUWDAHYGIOHS 10.8 Ki 2
QMCVFDPMIZPVDS 10.7 Ki 2
UWSVAGUSMAEUKO 10.7 Ki 2
ZQJBDIZBNGQJDT 10.6 Ki 2
SREQXWNZQCXRIR 10.6 Ki 2
AMNCJZAOSZGEBS 10.4 Ki 2
XVBGKELHGBXFDC 10.4 Ki 2
CTTYWAAVPCSYCV 10.4 Ki 2
HMBROJULWCDLQT 10.3 Ki 2
IPSNCGJWCSQSPB 10.3 Ki 2
JMCYOVXEMFWTCO 10.3 Ki 2
PHJUBIAVEOBIMZ 10.3 Ki 2
OVPADMIVRRGECP 10.3 Ki 2
JJPAWNWDPWKLCQ 10.3 Ki 2
SHDXBRHKJBXVOE 10.2 Ki 2
GNWGNQFZTKCMNP 10.2 Ki 2
ZQJBDIZBNGQJDT 10.2 Ki 2
LTVYROXJAPCACF 10.2 Ki 2
GSKRTNPTDULYSS 10.2 Ki 2
NYXKTTKEHKQLNH 10.1 Ki 2
OTLVIMXDRAAFAE 10.1 Ki 2
GVFUVCCZDCIYNB 10.1 Ki 2
BIPBOTWHSNMRCV 10.1 Ki 2
MSAPNOBIEOSWMP 10.1 Ki 2
CUFQBQOBLVLKRF 10.0 Ki 4
GKPIOXJPMSUIFL 10.0 Ki 2
RPIALZPTIFOQGC 10.0 Ki 3
NFLSBSNFRZFUJE 10.0 Ki 2
LNGFUEZUSQANCV 9.8 Ki 2
MPMUDVMRFYJRLP 9.8 Ki 2
QXISVZASIYAIRQ 9.8 Ki 2
ZQTXOGGDJIFYFB 9.8 Ki 2
LNGFUEZUSQANCV 9.8 Ki 2
LTSTXUQEHQNBBZ 9.8 Ki 2
RDGHXKOZJGWPHA 9.8 Ki 2
PAUIHFDXSPYWNF 9.7 Ki 2
LGCLJPYTRGJXHK 9.7 Ki 2
NHEIBOKBLUFHEF 9.7 Ki 2
QHMOOLGACYFYIQ 9.7 Ki 2
PGARSBKYUGXTLH 9.6 IC50 2
WWNPFAANLOAHOU 9.6 Ki 2
XGEGDSLAQZJGCW 9.6 Ki 2
WWNPFAANLOAHOU 9.6 Ki 2
UZLMEAPBHYEHAC 9.6 Ki 2
XCVGQMUMMDXKCY 9.6 Ki 3
LUZBHUHGIORDFL 9.6 Ki 2
2D structure