Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GNKSGLUNPBLOCF
|
7.0 | IC50 | 2 | — | |
JCGHBHWUCQLJPI
|
7.0 | IC50 | 2 | — | |
LOWZYNIZJZKVGV
|
7.0 | IC50 | 2 | — | |
MDIRLWZOKMHIJZ
|
7.0 | IC50 | 2 | — | |
WRJFIKUTCXERPD
|
7.0 | IC50 | 2 | — | |
CVKUHCDBBJWDLQ
|
7.0 | IC50 | 2 | — | |
SDDYKNWIADDTLB
|
7.0 | IC50 | 2 | — | |
JEORFMMREVWKES
|
6.9 | IC50 | 2 | — | |
JISVFSBNJCUDHU
|
6.9 | IC50 | 2 | — | |
NWGYHPLUCAMQRY
|
6.9 | IC50 | 2 | — | |
VRBHUDBHNQMOJO
|
6.9 | IC50 | 2 | — | |
VSEYNHJGEGEYBA
|
6.9 | IC50 | 2 | — | |
WGAFGKJZQIVWFL
|
6.9 | IC50 | 2 | — | |
QAVCQCQQTYJKSO
|
6.9 | IC50 | 2 | — | |
SVFKQHLOBRUZGV
|
6.9 | IC50 | 3 | — | |
CLJJLIVLJCOMDM
|
6.9 | IC50 | 2 | — | |
DFMUPSGOWRYRPS
|
6.9 | IC50 | 2 | — | |
IKITZJALQKJYEJ
|
6.9 | IC50 | 2 | — | |
KNXBMZUHMRSYTM
|
6.9 | IC50 | 2 | — | |
UPRAQJJHHIYMOB
|
6.9 | IC50 | 2 | — | |
IKZVNDBXJCSUFF
|
6.9 | IC50 | 2 | — | |
SSBKOEBEWJHUQR
|
6.9 | IC50 | 2 | — | |
AYCCBDPQSLELEH
|
6.9 | IC50 | 2 | — | |
OYXYUHYMXKMISB
|
6.9 | IC50 | 2 | — | |
UFLJTRYOECPADS
|
6.8 | IC50 | 2 | — | |
YYGQFCOCJWRYJT
|
6.8 | IC50 | 2 | — | |
INDZSXVDVYMLEE
|
6.8 | IC50 | 2 | — | |
OHJHLJNZRORZMK
|
6.8 | IC50 | 2 | — | |
PQQVQZLUXCWJBA
|
6.8 | IC50 | 2 | — | |
AGENJFMITVLRBS
|
6.8 | IC50 | 2 | — | |
CKKSVVDATCYHNV
|
6.8 | IC50 | 2 | — | |
YSEMEGXOKULCML
|
6.8 | IC50 | 2 | — | |
BERPEAVNCCSEPP
|
6.8 | IC50 | 2 | — | |
JFVMTILABAYJGC
|
6.8 | IC50 | 2 | — | |
BQBWWNAFFFKTGK
|
6.8 | IC50 | 2 | — | |
BBWJIFGPEJUGDS
|
6.8 | IC50 | 2 | — | |
HCXYAWFMXOIQEC
|
6.8 | IC50 | 2 | — | |
VLBKMGQYEGOGLA
|
6.8 | IC50 | 2 | — | |
BHJPHEXSIGFNTB
|
6.8 | IC50 | 2 | — | |
BOCZNEJOYWHXFD
|
6.8 | IC50 | 2 | — | |
FQLNOSMPZRXCRO
|
6.8 | IC50 | 2 | — | |
DMCPRSCBJQRXFA
|
6.8 | IC50 | 2 | — | |
FDYOAZVTGXEWGH
|
6.8 | IC50 | 2 | — | |
UJQMNATWMMSTAO
|
6.8 | IC50 | 2 | — | |
BJAUUCPOEAUGFQ
|
6.8 | IC50 | 2 | — | |
KAZIWSBVZDUBAI
|
6.7 | IC50 | 2 | — | |
KZBYGJHGWIMULJ
|
6.7 | IC50 | 2 | — | |
OPZYOXDFGXITFX
|
6.7 | IC50 | 2 | — | |
SOZVMXIKFABVBR
|
6.7 | IC50 | 2 | — | |
DEISFYWLJQPQHD
|
6.7 | IC50 | 2 | — |