Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BIKSKZHGVCCQDN
|
7.3 | IC50 | 2 | — | |
FLSSHCYZWNMCNZ
|
7.3 | IC50 | 2 | — | |
LZPSTBKXZZSDCN
|
7.3 | IC50 | 2 | — | |
PDGLHDNSYURVOE
|
7.3 | IC50 | 2 | — | |
GISQDTWWOXOIKD
|
7.3 | IC50 | 2 | — | |
WVVQRRCTXQZQNC
|
7.3 | IC50 | 2 | — | |
YSHVGBBWHQFDTL
|
7.3 | IC50 | 2 | — | |
OWQJVODOCWCIPX
|
7.2 | IC50 | 2 | — | |
SHONGYQWPMGFBR
|
7.2 | IC50 | 2 | — | |
SNKPYTPMXOONSA
|
7.2 | IC50 | 2 | — | |
LXKVZVZLCQFCKE
|
7.2 | IC50 | 2 | — | |
MDUVTBXIIMXLNO
|
7.2 | IC50 | 2 | — | |
ULVUURBFDYVMPY
|
7.2 | IC50 | 2 | — | |
YITDREASSSCOKM
|
7.2 | IC50 | 2 | — | |
SJNMBQBKAJVHAR
|
7.2 | IC50 | 2 | — | |
ITLJTFLFDKESMH
|
7.2 | IC50 | 2 | — | |
YAVWJVYAUHWKPJ
|
7.2 | IC50 | 2 | — | |
GOSIJUGDTWLDOF
|
7.2 | IC50 | 2 | — | |
LUYCFGBPBPYQHG
|
7.2 | IC50 | 2 | — | |
GKIQGOMXKXQVSO
|
7.2 | IC50 | 2 | — | |
CCJJPOCNADHZMF
|
7.2 | IC50 | 2 | — | |
IPVNHELRRJRWDT
|
7.2 | IC50 | 2 | — | |
LQQHADUYCCSZCE
|
7.2 | IC50 | 2 | — | |
RUFQBYAUEBPVOC
|
7.2 | IC50 | 2 | — | |
IOWSBZYCNNDVIQ
|
7.1 | IC50 | 2 | — | |
JWDXFZMJSOKLBM
|
7.1 | IC50 | 2 | — | |
ZBAIJDRMNLCRIN
|
7.1 | IC50 | 2 | — | |
GEJXMFWZAITGKE
|
7.1 | IC50 | 2 | — | |
GPYMFXQBCZGSRA
|
7.1 | IC50 | 2 | — | |
NQDJXKOVJZTUJA
|
7.1 | IC50 | 3 | — | |
QSEZKNHRUQRMIL
|
7.1 | IC50 | 2 | — | |
RMKJJNGAUVCDBG
|
7.1 | IC50 | 2 | — | |
PMXOHCADTKKKOM
|
7.1 | IC50 | 2 | — | |
CXJPWCNKFIWDQB
|
7.0 | IC50 | 2 | — | |
DUDOPGVSTUICEO
|
7.0 | IC50 | 2 | — | |
FPMFGCKVSAMYOU
|
7.0 | IC50 | 2 | — | |
KGODUAGFSYIJQW
|
7.0 | IC50 | 2 | — | |
NLDQVMDBRMGUMI
|
7.0 | IC50 | 2 | — | |
SGXFRGLRYZSEDC
|
7.0 | IC50 | 2 | — | |
XTZOFNNUVVUZHO
|
7.0 | IC50 | 2 | — | |
HHTVAFPSLHBBQG
|
7.0 | IC50 | 2 | — | |
HPKRLZZAMUMBAN
|
7.0 | IC50 | 2 | — | |
SQZJOEJUKUFRRK
|
7.0 | IC50 | 2 | — | |
AAWWSWAOXUPEEG
|
7.0 | IC50 | 2 | — | |
YVMOAVJHQOOGCA
|
7.0 | IC50 | 2 | — | |
BMCALDMFEXQQRY
|
7.0 | IC50 | 2 | — | |
GGICVMHKERQRRS
|
7.0 | IC50 | 2 | — | |
PJHNLYXCFFTMJX
|
7.0 | IC50 | 2 | — | |
ZQEDJHKILXMIFY
|
7.0 | IC50 | 2 | — | |
BFWCEJAASWLOBX
|
7.0 | IC50 | 2 | — |