Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JAHFQIYYIOEHDX
|
7.8 | IC50 | 2 | — | |
UEGXZQOTGTVUKD
|
7.8 | IC50 | 2 | — | |
XBXCMGXDWHDVNX
|
7.8 | IC50 | 2 | — | |
OSNHXMBZJPUQKF
|
7.7 | IC50 | 2 | — | |
KBVKZTXBAARIBF
|
7.7 | IC50 | 2 | — | |
MEDCPPNEGZYFET
|
7.7 | IC50 | 2 | — | |
OKBJYZHLIFUWOD
|
7.7 | IC50 | 2 | — | |
TYPYIAOCHCKFIA
|
7.7 | IC50 | 2 | — | |
UDDMNBYVRLYNKY
|
7.7 | IC50 | 2 | — | |
KPVDIIPFHYNTLD
|
7.7 | IC50 | 2 | — | |
MJMDFEZUPZGSHT
|
7.7 | IC50 | 2 | — | |
KLCNJQLRPTWZSY
|
7.7 | IC50 | 2 | — | |
AHAQASQWEHMCHG
|
7.6 | IC50 | 2 | — | |
KYDALGOIRAPGOG
|
7.6 | IC50 | 2 | — | |
IEESSKGGLUHWJD
|
7.6 | IC50 | 2 | — | |
BWPTVDYVVBUFBZ
|
7.6 | IC50 | 2 | — | |
FESKECLMGVLGFJ
|
7.6 | IC50 | 2 | — | |
UWBOVNUZRAIRLM
|
7.6 | IC50 | 2 | — | |
YZMDGUHXAPIFCJ
|
7.6 | IC50 | 2 | — | |
UYUIJOAWTJMMIV
|
7.6 | IC50 | 2 | — | |
WBEKDZJEFWTWEZ
|
7.6 | IC50 | 2 | — | |
KBNAVAPRJRYDCX
|
7.5 | IC50 | 2 | — | |
RGDXKPQBVYZPLJ
|
7.5 | IC50 | 2 | — | |
JTYHXCRYMXKNCE
|
7.5 | IC50 | 2 | — | |
OSCVHOFAXPMNHC
|
7.5 | IC50 | 2 | — | |
QTKKWORDBGQVCP
|
7.5 | IC50 | 2 | — | |
JMMPZYQZVRRZDH
|
7.5 | IC50 | 2 | — | |
CLDYKRBQBPQKDC
|
7.5 | IC50 | 2 | — | |
OWHAAVNYSQSALN
|
7.5 | IC50 | 2 | — | |
RIPOGUPNVLZOCZ
|
7.5 | IC50 | 2 | — | |
PVSSGUUFLHEGID
|
7.5 | IC50 | 2 | — | |
VIKCADRKXGMLKS
|
7.4 | IC50 | 2 | — | |
HDVZWQWXAQRFKJ
|
7.4 | IC50 | 3 | — | |
KJVILHBOZRFNJR
|
7.4 | IC50 | 2 | — | |
GSLBQKHXBYDHEM
|
7.4 | IC50 | 2 | — | |
QVBCGVSBAZFFCX
|
7.4 | IC50 | 2 | — | |
XWNJETQPIDITKR
|
7.4 | IC50 | 2 | — | |
ONXITTXWTWRVJA
|
7.4 | IC50 | 2 | — | |
IEZOLPNZJAVUST
|
7.4 | IC50 | 2 | — | |
KGWRKSLKDXAWRK
|
7.4 | IC50 | 2 | — | |
RBFYUIXVWQHOIR
|
7.4 | IC50 | 2 | — | |
PKICVKLKMOBLLB
|
7.4 | IC50 | 2 | — | |
FHJGAWQBOVTBCY
|
7.3 | IC50 | 2 | — | |
DGBVNIAUNCJNBL
|
7.3 | IC50 | 2 | — | |
ARXVVUNTVYPSIN
|
7.3 | IC50 | 2 | — | |
JKEVDPUWXLGMPH
|
7.3 | IC50 | 2 | — | |
GNMFKYCBSKMWKN
|
7.3 | IC50 | 2 | — | |
JYDIPPPAHISWJQ
|
7.3 | IC50 | 2 | — | |
UBIKZFFZJJPBBL
|
7.3 | IC50 | 2 | — | |
WUKFGTRLGMGCPE
|
7.3 | IC50 | 2 | — |