Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VXZGNFQKGJIROF
|
8.4 | IC50 | 2 | — | |
WESUQRYRDQAIIG
|
8.4 | IC50 | 2 | — | |
DVMRJJTXXYCAMY
|
8.4 | IC50 | 2 | — | |
ITNJYDYPEGKJNU
|
8.4 | IC50 | 2 | — | |
OKHSYOTXPAMJOC
|
8.4 | IC50 | 2 | — | |
OKHSYOTXPAMJOC
|
8.4 | IC50 | 2 | — | |
RDNNMGZPVVYTPG
|
8.4 | IC50 | 2 | — | |
XYWBREUGGXLQGJ
|
8.4 | IC50 | 2 | — | |
MOMJLJRBDDQQAF
|
8.3 | IC50 | 2 | — | |
ACIFBMIOXGVFDG
|
8.3 | IC50 | 2 | — | |
DOJWUCJRIDFBHM
|
8.3 | IC50 | 2 | — | |
DVMRJJTXXYCAMY
|
8.3 | IC50 | 2 | — | |
IGNUPIWYJJQPNO
|
8.3 | IC50 | 2 | — | |
IDXGOPPWFHQCNG
|
8.3 | IC50 | 2 | — | |
XQWXZKVWTDPJKP
|
8.3 | IC50 | 2 | — | |
UUCUKJOAGYJMSO
|
8.3 | IC50 | 2 | — | |
KLCNJQLRPTWZSY
|
8.3 | IC50 | 2 | — | |
QVPZFSZKKUMQOJ
|
8.3 | IC50 | 2 | — | |
YYHCGYHKXMRNOM
|
8.3 | IC50 | 2 | — | |
MSBCZCYTZAGQKP
|
8.3 | IC50 | 2 | — | |
WXNRGZGHPWMAKC
|
8.3 | IC50 | 2 | — | |
CTRVZTLOIONNSI
|
8.3 | IC50 | 2 | — | |
SCHMTZVKAUNPJE
|
8.3 | IC50 | 2 | — | |
CUMUAWSPWRJWGB
|
8.2 | IC50 | 2 | — | |
YJCRAEWURXHCGJ
|
8.2 | IC50 | 2 | — | |
PULATRQERYGHTK
|
8.2 | IC50 | 2 | — | |
FYYIANSYNMTNJP
|
8.2 | IC50 | 2 | — | |
HBVYIHSSCIKKFM
|
8.2 | IC50 | 2 | — | |
LHMFHMRJXAQDSO
|
8.2 | IC50 | 2 | — | |
KEOILRZETCFDMB
|
8.2 | IC50 | 2 | — | |
BFTAVSXREQVEFH
|
8.1 | IC50 | 2 | — | |
YEFVOKDOLXVJEU
|
8.1 | IC50 | 2 | — | |
YCRDKOUVJHLSMJ
|
8.1 | IC50 | 2 | — | |
QFWPUMZNHARHPP
|
8.1 | IC50 | 2 | — | |
AQODZPRBNVNXME
|
8.1 | IC50 | 2 | — | |
ITPSYHAKFLYHHN
|
8.1 | IC50 | 2 | — | |
LWFYAWCRFNADFC
|
8.1 | IC50 | 2 | — | |
CAMGSKZJCAYTIG
|
8.0 | IC50 | 2 | — | |
FHCWSFKYDKLLKL
|
8.0 | IC50 | 2 | — | |
PKTDOGBMTZCKJY
|
8.0 | IC50 | 2 | — | |
ZDUSJNCBGYSMMK
|
8.0 | IC50 | 2 | — | |
RKAFGUNUPCFFEF
|
8.0 | IC50 | 2 | — | |
KPLRYMADGNMCOA
|
8.0 | IC50 | 2 | — | |
YVVGGNNZPPNCKL
|
8.0 | IC50 | 2 | — | |
JQBBFMYGEYTZAB
|
7.9 | IC50 | 2 | — | |
JNNYBFVTFNQISB
|
7.9 | IC50 | 2 | — | |
XUMAZJDXZMTLHT
|
7.9 | IC50 | 2 | — | |
AVUMZHUUVRLIGV
|
7.9 | IC50 | 2 | — | |
UFHMRFDXZUEDFH
|
7.8 | IC50 | 2 | — | |
NUKQIBJIRBBHPZ
|
7.8 | IC50 | 2 | — |