Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HLMRLAVAJZMJRD
|
8.6 | IC50 | 2 | — | |
JQCHQBBQHKXONF
|
8.6 | IC50 | 2 | — | |
MUJZEQKONAELEN
|
8.6 | IC50 | 2 | — | |
NIGXLAOGARESRJ
|
8.6 | IC50 | 2 | — | |
OGMIECRJRAMAOQ
|
8.6 | IC50 | 2 | — | |
OTACRFHKBXUOMD
|
8.6 | IC50 | 2 | — | |
PBQBRNXINKAJFG
|
8.6 | IC50 | 2 | — | |
PWJRIHSLFKZKMA
|
8.6 | IC50 | 2 | — | |
QHCCRWMNOPPJSM
|
8.6 | IC50 | 2 | — | |
SNRKFDXIQAEWQI
|
8.6 | IC50 | 2 | — | |
SZWZZCQOINIKAI
|
8.6 | IC50 | 2 | — | |
TYQXZZJFCFIXDL
|
8.6 | IC50 | 2 | — | |
VBNAMCGXHGLJIT
|
8.6 | IC50 | 2 | — | |
VSNVAZOHAZBYGT
|
8.6 | IC50 | 2 | — | |
YRJUUGOXNJTWQU
|
8.6 | IC50 | 2 | — | |
YUDJDXATLXOJDR
|
8.6 | IC50 | 2 | — | |
ZHYCGZHKPUQEBV
|
8.6 | IC50 | 2 | — | |
ZOLIXMYUVIUJJN
|
8.6 | IC50 | 2 | — | |
BGLWBLAIIPWZRZ
|
8.5 | IC50 | 2 | — | |
GSBBITRNLVGMDT
|
8.5 | IC50 | 2 | — | |
HKSACYKKJSWVGC
|
8.5 | IC50 | 2 | — | |
JTIDGOJLNHZYPR
|
8.5 | IC50 | 2 | — | |
KIUGLMGWDVALJN
|
8.5 | IC50 | 2 | — | |
LHKPDMTVAOEUHM
|
8.5 | IC50 | 2 | — | |
LIFFFMXGDMHRIB
|
8.5 | IC50 | 2 | — | |
MYCXASANDFMMMO
|
8.5 | IC50 | 2 | — | |
OTYMNODPBXXNEZ
|
8.5 | IC50 | 2 | — | |
TUCPIXZXFYDFAP
|
8.5 | IC50 | 2 | — | |
WEJHEDBFTVRYIQ
|
8.5 | IC50 | 2 | — | |
ZGLWBLWOATZQFS
|
8.5 | IC50 | 2 | — | |
AWRQRQABLTZTPO
|
8.5 | IC50 | 2 | — | |
MGIGPVPBUCRTRQ
|
8.5 | IC50 | 2 | — | |
NXMUGBFAFCMFPR
|
8.5 | IC50 | 2 | — | |
QNKGCZRNGSRJSA
|
8.5 | IC50 | 2 | — | |
SDCWQJDGRJYYMI
|
8.5 | IC50 | 2 | — | |
VWMFQQRUWJOTHH
|
8.5 | IC50 | 2 | — | |
GMNKJWAVVVHELD
|
8.5 | IC50 | 2 | — | |
GWFBAUSRAWUPID
|
8.5 | IC50 | 2 | — | |
IKZPMPBBVSDQAT
|
8.5 | IC50 | 2 | — | |
PGPAAGCAINLZFM
|
8.5 | IC50 | 2 | — | |
WVRKVQIEEGRBRI
|
8.5 | IC50 | 2 | — | |
YHMQUWZYTCNQMT
|
8.5 | IC50 | 2 | — | |
CATYEFRZCMVTJK
|
8.5 | IC50 | 2 | — | |
FICOQFXHSFYJGJ
|
8.5 | IC50 | 2 | — | |
FZLHFGYEAHNEOS
|
8.5 | IC50 | 2 | — | |
GHJWZOWHDTUAPP
|
8.5 | IC50 | 2 | — | |
GUPAXIQAOINPLZ
|
8.5 | IC50 | 2 | — | |
HMFINSOGXKJQMS
|
8.5 | IC50 | 2 | — | |
HYJOGPCKSJXAQK
|
8.5 | IC50 | 2 | — | |
IVOVAMQTODMEAV
|
8.5 | IC50 | 2 | — |