Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LZRAXTRHYWUKJG
|
8.6 | IC50 | 2 | — | |
NFGZNHFRANDFII
|
8.6 | IC50 | 2 | — | |
OBDJMRKGTPYZKO
|
8.6 | IC50 | 2 | — | |
PHJCNYKEYZSING
|
8.6 | IC50 | 2 | — | |
QNKLZKKJTWWBIT
|
8.6 | IC50 | 2 | — | |
ZGKNNTCALNSSQV
|
8.6 | IC50 | 2 | — | |
CKCZUZAZTPNVOS
|
8.6 | IC50 | 2 | — | |
FYOQFKNCPYPJFT
|
8.6 | IC50 | 2 | — | |
GZWOTDFBINSOTK
|
8.6 | IC50 | 2 | — | |
HUZUWZSTVHYJLE
|
8.6 | IC50 | 2 | — | |
IOYHTOSBXCFLMW
|
8.6 | IC50 | 2 | — | |
MCPWYIAFNWICOU
|
8.6 | IC50 | 2 | — | |
NAWKKKKRFNMJTL
|
8.6 | IC50 | 2 | — | |
NEIMNGKOAGJOQH
|
8.6 | IC50 | 2 | — | |
NHCDEHMAKCLIEF
|
8.6 | IC50 | 2 | — | |
NTTJRCFSPLLJQO
|
8.6 | IC50 | 2 | — | |
OVSULEGCXRRXDG
|
8.6 | IC50 | 2 | — | |
QCUZUNFUUSLHHZ
|
8.6 | IC50 | 2 | — | |
QKRGGPXXHKITLQ
|
8.6 | IC50 | 2 | — | |
RJNQPEVMYJIZJN
|
8.6 | IC50 | 2 | — | |
UPIYQKNRYIWMJI
|
8.6 | IC50 | 2 | — | |
YHHUNANTYCEXPT
|
8.6 | IC50 | 2 | — | |
ZIODZEXPYWIBPG
|
8.6 | IC50 | 2 | — | |
BINKQGHRTGDRCO
|
8.6 | IC50 | 2 | — | |
CJXWTAGSUQXKFJ
|
8.6 | IC50 | 2 | — | |
FQUMQUZQLXOZSD
|
8.6 | IC50 | 2 | — | |
JHBQTJFLIQYZJE
|
8.6 | IC50 | 2 | — | |
JYSYRBLEEVBZMV
|
8.6 | IC50 | 2 | — | |
LKTBKLAVBLIIIS
|
8.6 | IC50 | 2 | — | |
OHDNVNJYYUPVKO
|
8.6 | IC50 | 2 | — | |
QHCCRWMNOPPJSM
|
8.6 | IC50 | 2 | — | |
RYGAGCQQONYYQS
|
8.6 | IC50 | 2 | — | |
TXERPEOOEKTJER
|
8.6 | IC50 | 2 | — | |
VEQZFJKYIWAJMO
|
8.6 | IC50 | 2 | — | |
YQJKAVNYWGMKFR
|
8.6 | IC50 | 2 | — | |
YXIUCOBYCBAULU
|
8.6 | IC50 | 2 | — | |
GILKVZODPWBBIF
|
8.6 | IC50 | 2 | — | |
HFWTVTRTAINKMO
|
8.6 | IC50 | 2 | — | |
JNSYXPGNGBSTBR
|
8.6 | IC50 | 2 | — | |
MNBCGSRAAVNTCP
|
8.6 | IC50 | 2 | — | |
NGUKEIRFKBTQGA
|
8.6 | IC50 | 2 | — | |
OFOCPMHFCFICDP
|
8.6 | IC50 | 2 | — | |
SFBZBTVMCAKLTJ
|
8.6 | IC50 | 2 | — | |
VSFISGOGKRGMSO
|
8.6 | IC50 | 2 | — | |
WOWIDUSMKYGEKX
|
8.6 | IC50 | 2 | — | |
ZRUAWOFGZUCGNA
|
8.6 | IC50 | 2 | — | |
CAJXCWZBDHKFDU
|
8.6 | IC50 | 2 | — | |
CXRSXNJDCNVSGA
|
8.6 | IC50 | 2 | — | |
DGLVSFSNOHORDG
|
8.6 | IC50 | 2 | — | |
GJANPMRITOIGHY
|
8.6 | IC50 | 2 | — |