Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WBWMIQNOMCEWQD
|
8.7 | IC50 | 2 | — | |
XVBYHQUWMKOCFW
|
8.7 | IC50 | 2 | — | |
XVBYHQUWMKOCFW
|
8.7 | IC50 | 2 | — | |
YODDPOMYGPZKCU
|
8.7 | IC50 | 2 | — | |
ZDUCWUQWVGUNPY
|
8.7 | IC50 | 2 | — | |
HLAFOQXZQAOOCA
|
8.7 | IC50 | 2 | — | |
LKVYUKUDUQXQSA
|
8.7 | IC50 | 2 | — | |
NSMSXEJRCLRXMM
|
8.7 | IC50 | 2 | — | |
OTUMQWWQYXWAOJ
|
8.7 | IC50 | 2 | — | |
OXQBEXIPUZDAMR
|
8.7 | IC50 | 2 | — | |
RCOJVGIUNNBVOW
|
8.7 | IC50 | 2 | — | |
SGKVBSKMQGODKO
|
8.7 | IC50 | 2 | — | |
ULLOSPYTXIBFQK
|
8.7 | IC50 | 2 | — | |
WPBWUFWECWKFMC
|
8.7 | IC50 | 2 | — | |
XRKGSRSDKJLMQO
|
8.7 | IC50 | 2 | — | |
XVBYHQUWMKOCFW
|
8.7 | IC50 | 2 | — | |
XVBYHQUWMKOCFW
|
8.7 | IC50 | 2 | — | |
ALQCKDCRKBPSFZ
|
8.7 | IC50 | 2 | — | |
CNNNYKMGCZBFEY
|
8.7 | IC50 | 2 | — | |
DWXUAYCYDSFTFG
|
8.7 | IC50 | 2 | — | |
FRJONNSVEZFPNQ
|
8.7 | IC50 | 2 | — | |
KOBIZTLMAWGBGX
|
8.7 | IC50 | 2 | — | |
LZFFMYMJKQUERJ
|
8.7 | IC50 | 2 | — | |
QSAZSARXXFUGPO
|
8.7 | IC50 | 2 | — | |
QWUUULZCSSEVQN
|
8.7 | IC50 | 2 | — | |
SKDPJVDWRZATOS
|
8.7 | IC50 | 2 | — | |
VOAWNBUAGRTURM
|
8.7 | IC50 | 2 | — | |
WFHWCFLWVVYTRJ
|
8.7 | IC50 | 2 | — | |
YORLWSMAYZWBLB
|
8.7 | IC50 | 2 | — | |
ZOKBZRIQVNLAEX
|
8.7 | IC50 | 2 | — | |
NTTJRCFSPLLJQO
|
8.7 | IC50 | 2 | — | |
ADNLZSHYYLCKRF
|
8.6 | IC50 | 2 | — | |
IADAQZBFGHOPKF
|
8.6 | IC50 | 2 | — | |
IEPKYTYVGHEUOE
|
8.6 | IC50 | 2 | — | |
KVHGELDGJLZSQB
|
8.6 | IC50 | 2 | — | |
LTTDWRSUTZHAAM
|
8.6 | IC50 | 2 | — | |
MLEXGMXFORMIDH
|
8.6 | IC50 | 2 | — | |
OTKJRMPQQAZWAM
|
8.6 | IC50 | 2 | — | |
PVHLNTJIIZEGRI
|
8.6 | IC50 | 2 | — | |
QTCOSGLPXCDGIR
|
8.6 | IC50 | 2 | — | |
SHHRLXAXOOHOES
|
8.6 | IC50 | 2 | — | |
VZIBQPOBCHDMRZ
|
8.6 | IC50 | 2 | — | |
WIDJQXBMYMMVAB
|
8.6 | IC50 | 2 | — | |
ZYCWGMRUIYKCFU
|
8.6 | IC50 | 2 | — | |
ACXWAWUMTPBWBX
|
8.6 | IC50 | 2 | — | |
CIOCDOCQXNPPAP
|
8.6 | IC50 | 2 | — | |
CYMPINQHDXGKOA
|
8.6 | IC50 | 2 | — | |
FRIDTZAQHLGVTN
|
8.6 | IC50 | 2 | — | |
HJJCAAZJYRMDJK
|
8.6 | IC50 | 2 | — | |
IEGCCNRDFHUOGM
|
8.6 | IC50 | 2 | — |